| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA920099 | F | Trypanocidal activity against Trypanosoma cruzi Y blood stream trypomastigotes assessed as parasite lysis at 0.31 mM relative to control | Trypanosoma cruzi | 8 | ALA1144512 | organism-based format | Scientific Literature | |
| 2. | ALA920100 | F | Trypanocidal activity against Trypanosoma cruzi Y blood stream trypomastigotes assessed as parasite lysis at 0.63 mM relative to control | Trypanosoma cruzi | 8 | ALA1144512 | organism-based format | Scientific Literature | |
| 3. | ALA920101 | F | Trypanocidal activity against Trypanosoma cruzi Y blood stream trypomastigotes assessed as parasite lysis at 1.25 mM relative to control | Trypanosoma cruzi | 7 | ALA1144512 | organism-based format | Scientific Literature | |
| 4. | ALA920102 | F | Trypanocidal activity against Trypanosoma cruzi Y blood stream trypomastigotes assessed as parasite lysis at 2.50 mM relative to control | Trypanosoma cruzi | 8 | ALA1144512 | organism-based format | Scientific Literature | |
| 5. | ALA920103 | F | Trypanocidal activity against blood stream Trypanosoma cruzi Y trypomastigotes assessed as parasite lysis at 5 mM relative to control | Trypanosoma cruzi | 8 | ALA1144512 | organism-based format | Scientific Literature | |
| 6. | ALA965909 | A | Growth inhibition of mouse L929 cells | Mus musculus | 11 | ALA1148912 | cell-based format | Scientific Literature | |
| 7. | ALA965910 | F | Growth inhibition of human K562 cells | Homo sapiens | 11 | ALA1148912 | cell-based format | Scientific Literature | |
| 8. | ALA965911 | F | Cytotoxicity against human HeLa cells | Homo sapiens | 11 | ALA1148912 | cell-based format | Scientific Literature | |
| 9. | ALA986772 | F | Antiviral activity against HIV1 3B replication in human H9 cells up to 100 ug/mL after 3 days by p24 antigen capture assay | Human immunodeficiency virus 1 | 12 | ALA1158287 | organism-based format | Scientific Literature | |
| 10. | ALA975593 | B | Inhibition of HIV reverse transcriptase at 33 ug/mL by scintillation counting | Human immunodeficiency virus | 4 | ALA1158673 | assay format | Scientific Literature | |
| 11. | ALA2405915 | B | Inhibition of mouse 11beta-HSD1 expressed in HEK293 cell microsomes assessed as inhibition of [3H]cortisone conversion to [3H]cortisol at 1 uM by scintillation proximity assay | Mus musculus | 39 | ALA2401669 | microsome format | Scientific Literature | |
| 12. | ALA2405916 | B | Inhibition of human 11beta-HSD1 expressed in HEK293 cell microsomes assessed as inhibition of [3H]cortisone conversion to [3H]cortisol at 1 uM by scintillation proximity assay | Homo sapiens | 39 | ALA2401669 | microsome format | Scientific Literature | |
| 13. | ALA2405917 | B | Inhibition of human 11beta-HSD2 | Homo sapiens | 15 | ALA2401669 | single protein format | Scientific Literature | |
| 14. | ALA2405918 | B | selectivity ratio of IC50 for human 11beta-HSD2 to IC50 for human 11beta-HSD1 | Homo sapiens | 15 | ALA2401669 | assay format | Scientific Literature | |
| 15. | ALA2405919 | B | Inhibition of human 11beta-HSD1 expressed in HEK293 cell microsomes assessed as inhibition of [3H]cortisone conversion to [3H]cortisol by scintillation proximity assay | Homo sapiens | 15 | ALA2401669 | microsome format | Scientific Literature | |
| 16. | ALA2405920 | B | Inhibition of mouse 11beta-HSD1 expressed in HEK293 cell microsomes assessed as inhibition of [3H]cortisone conversion to [3H]cortisol by scintillation proximity assay | Mus musculus | 15 | ALA2401669 | microsome format | Scientific Literature | |
| 17. | ALA2405921 | B | Inhibition of mouse 11beta-HSD2 | Mus musculus | 15 | ALA2401669 | single protein format | Scientific Literature | |
| 18. | ALA2405922 | B | Selectivity ratio of IC50 for mouse 11beta-HSD2 to IC50 for mouse 11beta-HSD1 | Mus musculus | 15 | ALA2401669 | assay format | Scientific Literature |
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