| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA1022735 | B | Inhibition of IGF1R | 25 | single protein format | Scientific Literature | |||
| 2. | ALA1022736 | B | Inhibition of IGF1R in mouse SAL cells assessed as thymidine incorporation | Mus musculus | 25 | cell-based format | Scientific Literature | ||
| 3. | ALA1022737 | A | Inhibition of CYP3A4 | 25 | single protein format | Scientific Literature | |||
| 4. | ALA1022738 | A | AUC (0 to 4 hrs) in mouse plasma at 20 mg/kg, po | Mus musculus | 24 | organism-based format | Scientific Literature | ||
| 5. | ALA1022739 | A | Metabolic stability in mouse liver microsomes | Mus musculus | 20 | microsome format | Scientific Literature | ||
| 6. | ALA1102236 | B | Inhibition of human recombinant IGF-1R tyrosine kinase expressed in baculovirus system assessed as [33gamma]ATP phosphorylation of poly(Glu/Tyr) substrate after 45 mins by scintillation counting | Homo sapiens | 34 | assay format | Scientific Literature | ||
| 7. | ALA1102237 | B | Transactivation activity at human PXR assessed as induction of CYP3A4 activity at 10 uMol/l relative to rifampicin | Homo sapiens | 34 | single protein format | Scientific Literature | ||
| 8. | ALA1102238 | A | Inhibition of CYP3A4 after 20 mins by BFC fluorescence assay | 17 | single protein format | Scientific Literature |
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