| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA995584 | B | Inhibition of human 11beta HSD1 by SPA assay | Homo sapiens | 52 | ALA1150311 | single protein format | Scientific Literature | |
| 2. | ALA995585 | B | Inhibition of mouse 11beta HSD1 by SPA assay | Mus musculus | 52 | ALA1150311 | single protein format | Scientific Literature | |
| 3. | ALA995589 | F | Inhibition of [3H]cortisone to [3H]cortisol conversion in mouse at 10 mg/kg, po administered as single dose after 4 hrs | Mus musculus | 36 | ALA1150311 | organism-based format | Scientific Literature | |
| 4. | ALA995590 | F | Inhibition of [3H]cortisone to [3H]cortisol conversion in mouse at 10 mg/kg, po administered as single dose after 16 hrs | Mus musculus | 13 | ALA1150311 | organism-based format | Scientific Literature | |
| 5. | ALA995591 | F | Agonist activity at human PXR | Homo sapiens | 15 | ALA1150311 | assay format | Scientific Literature | |
| 6. | ALA5246988 | B | Activation of PXR in human HepG2 cells at 1 uM incubated for 48 hrs relative to rifampicin | Homo sapiens | 4 | ALA5244274 | cell-based format | Scientific Literature | |
| 7. | ALA5246989 | B | Activation of PXR in human HepG2 cells at 10 uM incubated for 48 hrs relative to rifampicin | Homo sapiens | 4 | ALA5244274 | cell-based format | Scientific Literature | |
| 8. | ALA5246990 | A | Induction of CYP3A4 in human hepatocytes assessed as fold increase in mRNA level at 10 uM | Homo sapiens | 4 | ALA5244274 | cell-based format | Scientific Literature | |
| 9. | ALA5246991 | B | Inhibition of human 11beta-HSD1 | Homo sapiens | 4 | ALA5244274 | single protein format | Scientific Literature | |
| 10. | ALA5246992 | B | Activation of PXR (unknown origin) | Homo sapiens | 12 | ALA5244274 | single protein format | Scientific Literature |
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