# | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
---|---|---|---|---|---|---|---|---|---|
1. | ALA994997 | Functional | Antagonist activity at 5HT6 receptor expressed in HeLa cells assessed as 5HT-induced cAMP accumulation by chemiluminescence assay | 12 | ALA1144232 | cell-based format | Scientific Literature | ||
2. | ALA994998 | ADME | Metabolic stability in rat liver microsomes assessed as intrinsic clearance at 2 mM upto 30 mins | Rattus norvegicus | 12 | ALA1144232 | microsome format | Scientific Literature | |
3. | ALA995002 | ADME | Inhibition of human CYP3A4 by microtiter plate assays using N-N,diethyl-formamide as substrate | Homo sapiens | 12 | ALA1144232 | single protein format | Scientific Literature | |
4. | ALA995004 | Functional | Antagonist activity at 5HT2A receptor | 1 | ALA1144232 | assay format | Scientific Literature | ||
5. | ALA995005 | Functional | Antagonist activity at 5HT2B receptor | 1 | ALA1144232 | assay format | Scientific Literature | ||
6. | ALA995006 | Functional | Antagonist activity at 5HT2C receptor | 1 | ALA1144232 | assay format | Scientific Literature | ||
7. | ALA995007 | Binding | Ex vivo displacement of [125I]258585 from 5HT6 receptor in po dosed rat striatum | Rattus norvegicus | 1 | ALA1144232 | organism-based format | Scientific Literature | |
8. | ALA991619 | ADME | Inhibition of human CYP3A4 by microtiter plate assays using PPR substrate | Homo sapiens | 12 | ALA1144232 | single protein format | Scientific Literature |