| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA1000644 | B | Displacement of [3H]diprenorphine from human cloned kappa opioid receptor by cell based assay | Homo sapiens | 22 | ALA1136971 | cell-based format | Scientific Literature | |
| 2. | ALA1000645 | B | Displacement of [3H]diprenorphine from human cloned mu receptor by cell based assay | Homo sapiens | 22 | ALA1136971 | cell-based format | Scientific Literature | |
| 3. | ALA1000646 | B | Displacement of [3H]diprenorphine from human cloned delta receptor by cell based assay | Homo sapiens | 22 | ALA1136971 | cell-based format | Scientific Literature | |
| 4. | ALA1000647 | B | Ratio of Ki for human cloned mu opioid receptor to Ki for human cloned kappa opioid receptor | Homo sapiens | 13 | ALA1136971 | assay format | Scientific Literature | |
| 5. | ALA1000648 | F | Antagonist activity at human cloned kappa opioid receptor assessed as inhibition of 50 nM U50488H-stimulated GTPgammaS binding by cell based assay | Homo sapiens | 22 | ALA1136971 | cell-based format | Scientific Literature | |
| 6. | ALA1000649 | F | Antagonist activity at human cloned mu opioid receptor assessed as inhibition of 100 nM loperamide-stimulated GTPgammaS binding by cell based assay | Homo sapiens | 22 | ALA1136971 | cell-based format | Scientific Literature | |
| 7. | ALA2327127 | F | Antinociceptive activity in C57B1/6J mouse at 10 nmol, icv administered 80 mins prior to U50488 addition by warm water tail withdrawal assay | Mus musculus | 1 | ALA2321730 | organism-based format | Scientific Literature | |
| 8. | ALA2327130 | F | Inhibition of dynorphin A (1-13) NH2 binding to rat cloned KOR by [35S]GTPgammaS binding assay | Rattus norvegicus | 1 | ALA2321730 | assay format | Scientific Literature | |
| 9. | ALA2327131 | B | Displacement of [3H]DAMGO from rat cloned MOR expressed in CHO cells after 90 mins by scintillation counting analysis | Rattus norvegicus | 2 | ALA2321730 | cell-based format | Scientific Literature | |
| 10. | ALA2327132 | B | Displacement of [3H]DPDPE from mouse cloned DOR expressed in CHO cells after 90 mins by scintillation counting analysis | Mus musculus | 2 | ALA2321730 | cell-based format | Scientific Literature | |
| 11. | ALA2327133 | B | Displacement of [3H]diprenorphine from rat cloned KOR expressed in CHO cells after 90 mins by scintillation counting analysis | Rattus norvegicus | 2 | ALA2321730 | cell-based format | Scientific Literature | |
| 12. | ALA5127613 | B | Displacement of [3H]DAMGO from rat MOP stably expressed in CHO cell membrane | Rattus norvegicus | 6 | ALA5126521 | cell membrane format | Scientific Literature | |
| 13. | ALA5127614 | B | Displacement of [3H]DPDPE from mouse DOP stably expressed in CHO cell membrane | Mus musculus | 5 | ALA5126521 | cell membrane format | Scientific Literature | |
| 14. | ALA5127615 | B | Displacement of [3H]diprenorphine from rat KOP stably expressed in CHO cell membrane | Rattus norvegicus | 6 | ALA5126521 | cell membrane format | Scientific Literature | |
| 15. | ALA5127616 | B | Binding affinity to human KOP stably expressed in CHO cell membrane assessed as [35S]GTPgammaS binding | Homo sapiens | 2 | ALA5126521 | cell membrane format | Scientific Literature | |
| 16. | ALA5127624 | F | Antinociceptive activity in po dosed C57BL/6J mouse assessed as tail withdrawal latency from warm water | Mus musculus | 4 | ALA5126521 | organism-based format | Scientific Literature |
The page will load shortly, Thanks for your patience!