| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA973552 | B | Displacement of [3H]2-BFI from Imidazoline receptor 2 in Sprague-Dawley rat whole brain membrane | Rattus norvegicus | 12 | assay format | Scientific Literature | ||
| 2. | ALA973553 | B | Displacement of [3H]RX821002 from Adrenergic alpha2 receptor in Sprague-Dawley rat whole brain membrane | Rattus norvegicus | 12 | assay format | Scientific Literature | ||
| 3. | ALA973554 | B | Selectivity ratio, IC50 for Imidazoline receptor 1 in Sprague-Dawley rat kidney membrane to Ki for Imidazoline receptor 2 in Sprague-Dawley rat whole brain membrane | Rattus norvegicus | 12 | cell membrane format | Scientific Literature | ||
| 4. | ALA973555 | B | Selectivity ratio, IC50 for Imidazoline receptor 1 in Sprague-Dawley rat kidney membrane to Ki for alpha2 adrenoceptor in Sprague-Dawley rat whole brain membrane | Rattus norvegicus | 12 | cell membrane format | Scientific Literature | ||
| 5. | ALA973556 | B | Displacement of [3H]clonidine from Imidazoline receptor 1 rat PC-12 cells | Rattus norvegicus | 2 | cell-based format | Scientific Literature | ||
| 6. | ALA973557 | B | Binding affinity to Imidazoline receptor 2 | 2 | assay format | Scientific Literature | |||
| 7. | ALA973558 | B | Selectivity ratio, pKi for Imidazoline receptor 2 to pKi for Imidazoline receptor 1 | 2 | assay format | Scientific Literature | |||
| 8. | ALA973559 | B | Selectivity ratio, pKi for Imidazoline receptor 2 to pKi for alpha2 adrenoceptor | 2 | assay format | Scientific Literature | |||
| 9. | ALA973562 | F | Decrease in morphine-induced analgesia in CD1 mouse at 10 mg/kg, sc after 30 mins by tail flick test relative to control | Mus musculus | 5 | organism-based format | Scientific Literature | ||
| 10. | ALA973565 | F | Effect on morphine-induced analgesia in yohimbine pretreated CD1 mouse at 10 mg/kg, sc by tail flick test | Mus musculus | 2 | organism-based format | Scientific Literature | ||
| 11. | ALA973566 | F | Effect on morphine-induced analgesia in efaroxan pretreated CD1 mouse at 10 mg/kg, sc by tail flick test | Mus musculus | 2 | organism-based format | Scientific Literature | ||
| 12. | ALA968879 | F | Reversal of decrease in morphine-induced analgesia in idazoxan pretreated CD1 mouse at 10 mg/kg, sc by tail flick assay | Mus musculus | 2 | organism-based format | Scientific Literature | ||
| 13. | ALA3056380 | B | Binding affinity to I2 imidazoline binding site (unknown origin) | Homo sapiens | 25 | assay format | Scientific Literature | ||
| 14. | ALA3056381 | B | Binding affinity to I1 imidazoline binding site in Rattus norvegicus (rat) PC12 cells | Rattus norvegicus | 25 | cell-based format | Scientific Literature |
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