| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA997028 | Binding | Inhibition of human recombinant cathepsin S by fluorometric assay | Homo sapiens | 23 | ALA1156562 | single protein format | Scientific Literature | |
| 2. | ALA997029 | Binding | Inhibition of human recombinant cathepsin K by fluorometric assay | Homo sapiens | 14 | ALA1156562 | single protein format | Scientific Literature | |
| 3. | ALA997030 | Binding | Inhibition of human recombinant cathepsin L by fluorometric assay | Homo sapiens | 23 | ALA1156562 | single protein format | Scientific Literature | |
| 4. | ALA997031 | Binding | Selectivity for human recombinant cathepsin S over human recombinant cathepsin L | Homo sapiens | 4 | ALA1156562 | assay format | Scientific Literature | |
| 5. | ALA997032 | Physicochemical | Aqueous solubility at pH 6.8 | 4 | ALA1156562 | small-molecule physicochemical format | Scientific Literature | ||
| 6. | ALA997033 | ADME | Clearance in Sprague-Dawley rat at 1 mg/kg, iv and 3 mg/kg, po | Rattus norvegicus | 3 | ALA1156562 | organism-based format | Scientific Literature | |
| 7. | ALA997035 | ADME | Half life in Sprague-Dawley rat at 1 mg/kg, iv | Rattus norvegicus | 4 | ALA1156562 | organism-based format | Scientific Literature | |
| 8. | ALA997036 | ADME | Bioavailability in Sprague-Dawley rat at 1 mg/kg, iv and 3 mg/kg, po | Rattus norvegicus | 3 | ALA1156562 | organism-based format | Scientific Literature | |
| 9. | ALA997038 | ADME | Normalized AUC in Sprague-Dawley rat at 1 mg/kg, po | Rattus norvegicus | 4 | ALA1156562 | organism-based format | Scientific Literature | |
| 10. | ALA997039 | Binding | Inhibition of cathepsin S in mouse A20 cells assessed as invariant chain degradation at 1 uM | Mus musculus | 3 | ALA1156562 | cell-based format | Scientific Literature |
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