| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA1827029 | B | Binding affinity to H4R receptor | 2 | single protein format | Scientific Literature | |||
| 2. | ALA1827030 | B | Inhibition of 5-HT3AR at 10 uM | 2 | single protein format | Scientific Literature | |||
| 3. | ALA948406 | F | Antagonist activity at human histamine H4 receptor expressed in HEK293 cells coexpressing G-protein assessed as inhibition of histamine-induced intracellular calcium level by FLIPR | Homo sapiens | 2 | cell-based format | Scientific Literature | ||
| 4. | ALA948407 | F | Antagonist activity at rat histamine H4 receptor assessed as inhibition of histamine-induced intracellular calcium level by FLIPR | Rattus norvegicus | 2 | cell-based format | Scientific Literature | ||
| 5. | ALA948408 | F | Antagonist activity at mouse histamine H4 receptor assessed as inhibition of histamine-induced intracellular calcium level by FLIPR | Mus musculus | 2 | cell-based format | Scientific Literature | ||
| 6. | ALA948409 | F | Antagonist activity at rat histamine H4 receptor assessed as inhibition of histamine-induced [35S]GTPgamma binding | Rattus norvegicus | 1 | assay format | Scientific Literature | ||
| 7. | ALA948410 | B | Displacement of [3H]histamine from human histamine H4 receptor expressed in HEK293 cells by liquid scintillation counting | Homo sapiens | 2 | cell-based format | Scientific Literature | ||
| 8. | ALA948411 | B | Displacement of [3H]histamine from rat histamine H4 receptor expressed in HEK293 cells by liquid scintillation counting | Rattus norvegicus | 2 | cell-based format | Scientific Literature | ||
| 9. | ALA948412 | B | Binding affinity to human histamine H1 receptor | Homo sapiens | 2 | single protein format | Scientific Literature | ||
| 10. | ALA951435 | B | Binding affinity to human histamine H2 receptor | Homo sapiens | 2 | single protein format | Scientific Literature | ||
| 11. | ALA951436 | B | Binding affinity to human histamine H3 receptor | Homo sapiens | 2 | single protein format | Scientific Literature | ||
| 12. | ALA951437 | B | Binding affinity to rat histamine H3 receptor | Rattus norvegicus | 2 | single protein format | Scientific Literature | ||
| 13. | ALA951438 | A | Bioavailability in Sprague-Dawley rat at 10 mg/kg, ip | Rattus norvegicus | 1 | organism-based format | Scientific Literature | ||
| 14. | ALA951439 | A | Half life in Sprague-Dawley rat at 10 mg/kg, ip | Rattus norvegicus | 1 | organism-based format | Scientific Literature | ||
| 15. | ALA951440 | A | Cmax in Sprague-Dawley rat at 10 mg/kg, ip | Rattus norvegicus | 1 | organism-based format | Scientific Literature | ||
| 16. | ALA951441 | A | Tmax in Sprague-Dawley rat at 10 mg/kg, ip | Rattus norvegicus | 1 | organism-based format | Scientific Literature | ||
| 17. | ALA951442 | A | Oral bioavailability in Sprague-Dawley rat at 10 mg/kg | Rattus norvegicus | 1 | organism-based format | Scientific Literature | ||
| 18. | ALA951443 | A | Half life in Sprague-Dawley rat at 10 mg/kg, po | Rattus norvegicus | 1 | organism-based format | Scientific Literature | ||
| 19. | ALA951444 | A | Cmax in Sprague-Dawley rat at 10 mg/kg, po | Rattus norvegicus | 1 | organism-based format | Scientific Literature | ||
| 20. | ALA951445 | A | Tmax in Sprague-Dawley rat at 10 mg/kg, po | Rattus norvegicus | 1 | organism-based format | Scientific Literature |
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