# | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
---|---|---|---|---|---|---|---|---|---|
1. | ALA3791346 | Functional | Agonist activity at human FFA1 receptor expressed in human 1321N1 cells measured for 50 intervals of 0.4 secs by calcium mobilization assay | Homo sapiens | 19 | ALA3785041 | cell-based format | Scientific Literature | |
2. | ALA3791347 | Functional | Agonist activity at human FFA1 receptor expressed in human 1321N1 cells measured for 50 intervals of 0.4 secs by calcium mobilization assay relative to TUG-20 | Homo sapiens | 16 | ALA3785041 | cell-based format | Scientific Literature | |
3. | ALA3791350 | Binding | Agonist activity at human C-terminal YFP-tagged FFA4 receptor expressed in HEK293 cells incubated for 5 mins by BRET based beta-arrestin 2 recruitment assay | Homo sapiens | 18 | ALA3785041 | cell-based format | Scientific Literature | |
4. | ALA3791351 | Binding | Agonist activity at human C-terminal YFP-tagged FFA4 receptor expressed in HEK293 cells incubated for 5 mins by BRET based beta-arrestin 2 recruitment assay relative to TUG-424 | Homo sapiens | 11 | ALA3785041 | cell-based format | Scientific Literature | |
5. | ALA1775298 | Functional | Agonist activity at human FFA1 transfected in 1321N1 cells assessed as calcium mobilization by microplate assay | Homo sapiens | 33 | ALA1773039 | cell-based format | Scientific Literature | |
6. | ALA1775299 | Functional | Agonist activity at human FFA1 transfected in 1321N1 cells assessed as calcium mobilization by microplate assay relative to 10 uM TUG-20 | Homo sapiens | 32 | ALA1773039 | cell-based format | Scientific Literature | |
7. | ALA1775302 | Binding | Transactivation of human PPARgamma ligand binding domain transfected in mouse embryo fibroblasts assessed as renilla luciferase activity at 1 uM after 18 hrs by luminometry relative to 1 uM rosiglitazone | Homo sapiens | 31 | ALA1773039 | assay format | Scientific Literature | |
8. | ALA1775303 | Binding | Selectivity for human FFA1 over human PPARgamma | Homo sapiens | 30 | ALA1773039 | assay format | Scientific Literature | |
9. | ALA1775395 | Functional | Agonist activity at human GPR43 in HEK293 cells | Homo sapiens | 31 | ALA1773039 | cell-based format | Scientific Literature | |
10. | ALA1775396 | Functional | Agonist activity at human GPR41 in HEK293 cells | Homo sapiens | 31 | ALA1773039 | cell-based format | Scientific Literature | |
11. | ALA1833690 | Functional | Agonist activity at human FFA1 receptor expressed in human 1321N1 cells assessed as calcium mobilization by fluorescence spectrophotometry | Homo sapiens | 40 | ALA1828561 | cell-based format | Scientific Literature | |
12. | ALA1833691 | Functional | Agonist activity at human FFA1 receptor expressed in human 1321N1 cells assessed as calcium mobilization by fluorescence spectrophotometry relative to 10 uM TUG-20 | Homo sapiens | 33 | ALA1828561 | cell-based format | Scientific Literature | |
13. | ALA949441 | Functional | Agonist activity at human FFA1 expressed in human 1321N1 cells by calcium fluorescence assay | Homo sapiens | 18 | ALA1152274 | cell-based format | Scientific Literature | |
14. | ALA949443 | Functional | Agonist activity at human FFA1 expressed in human 1321N1 cells by calcium fluorescence assay relative to 3-(4-(benzyloxy)phenyl)propionic acid | Homo sapiens | 18 | ALA1152274 | cell-based format | Scientific Literature | |
15. | ALA949445 | Functional | Agonist activity at FFA2 | 21 | ALA1152274 | assay format | Scientific Literature | ||
16. | ALA949446 | Functional | Agonist activity at FFA3 | 21 | ALA1152274 | assay format | Scientific Literature | ||
17. | ALA2389877 | Binding | Agonist activity at C-terminal yellow fluorescent protein-fused human FFA4 receptor transfected in HEK293 cells after 5 mins by BRET assay relative to TUG-424 | Homo sapiens | 16 | ALA2384913 | cell-based format | Scientific Literature | |
18. | ALA2389878 | Functional | Agonist activity at human FFA1 receptor transfected in human 1321N1 cells by calcium mobilization assay relative to TUG-20 | Homo sapiens | 22 | ALA2384913 | cell-based format | Scientific Literature | |
19. | ALA2389879 | Binding | Agonist activity at C-terminal yellow fluorescent protein-fused human FFA4 receptor transfected in HEK293 cells after 5 mins by BRET assay | Homo sapiens | 22 | ALA2384913 | cell-based format | Scientific Literature | |
20. | ALA2389880 | Functional | Agonist activity at human FFA1 receptor transfected in human 1321N1 cells by calcium mobilization assay | Homo sapiens | 22 | ALA2384913 | cell-based format | Scientific Literature |