# | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
---|---|---|---|---|---|---|---|---|---|
1. | ALA946271 | B | Inhibition of 2-oxoglutarate-dependent human JMJD2E in presence of excess 2-oxoglutarate and 10 uM Fe2 by FDH coupled assay | Homo sapiens | 18 | ALA1152272 | assay format | Scientific Literature | |
2. | ALA946272 | B | Inhibition of 2-oxoglutarate-dependent human JMJD2E in presence of excess H3K9me3 peptide and 10 uM Fe2 by FDH coupled assay | Homo sapiens | 18 | ALA1152272 | assay format | Scientific Literature | |
3. | ALA946273 | B | Inhibition of 2-oxoglutarate-dependent human JMJD2E preincubated for 30 mins by FDH coupled assay | Homo sapiens | 13 | ALA1152272 | assay format | Scientific Literature | |
4. | ALA946281 | B | Inhibition of 2-oxoglutarate-dependent human recombinant HIF PHD2 preincubated for 1 hr | Homo sapiens | 2 | ALA1152272 | single protein format | Scientific Literature | |
5. | ALA1006265 | B | Inhibition of human recombinant PHD2 (181-426) expressed in Escherichia coli BL21 (DE3) by TR-FRET assay | Homo sapiens | 8 | ALA1138478 | assay format | Scientific Literature | |
6. | ALA1006266 | B | Destabilizing effect on human recombinant PHD2 (181-426) expressed in Escherichia coli BL21 (DE3) assessed as half life by limited trypsinolysis/MALDI-MS analysis in presence of ferrous ion | Homo sapiens | 7 | ALA1138478 | assay format | Scientific Literature | |
7. | ALA1008236 | B | Inhibition of mouse Oat6-mediated [3H]ES uptake in Xenopus oocytes after 1 hr | Mus musculus | 45 | ALA1156472 | cell-based format | Scientific Literature | |
8. | ALA1008237 | B | Inhibition of mouse Oat1-mediated [3H]PAH uptake in Xenopus oocytes after 1 hr | Mus musculus | 45 | ALA1156472 | cell-based format | Scientific Literature | |
9. | ALA1008238 | B | Ratio of pKi for mouse Oat1 expressed in Xenopus oocytes to pKi for mouse Oat6 expressed in Xenopus oocytes | Mus musculus | 45 | ALA1156472 | cell-based format | Scientific Literature | |
10. | ALA1053226 | B | Activation of human recombinant wild type mitochondrial NADP-ME expressed in Escherichia coli BL21 assessed as one-half maximal activation by spectrophotometry | Homo sapiens | 2 | ALA1153457 | assay format | Scientific Literature | |
11. | ALA1053227 | B | Activation of human mitochondrial NADP-ME E59L mutant expressed in Escherichia coli XL-1 by spectrophotometry | Homo sapiens | 1 | ALA1153457 | assay format | Scientific Literature | |
12. | ALA1068060 | B | Inhibition of human recombinant carbonic anhydrase 2 by stopped flow CO2 hydration method | Homo sapiens | 30 | ALA1157705 | single protein format | Scientific Literature | |
13. | ALA1068061 | B | Inhibition of human recombinant carbonic anhydrase 1 by stopped flow CO2 hydration method | Homo sapiens | 30 | ALA1157705 | single protein format | Scientific Literature | |
14. | ALA1068062 | B | Inhibition of human recombinant carbonic anhydrase 5A by stopped flow CO2 hydration method | Homo sapiens | 30 | ALA1157705 | single protein format | Scientific Literature | |
15. | ALA1068063 | B | Inhibition of human recombinant carbonic anhydrase 5B by stopped flow CO2 hydration method | Homo sapiens | 30 | ALA1157705 | single protein format | Scientific Literature | |
16. | ALA1068064 | B | Selectivity ratio of Kinact for human recombinant carbonic anhydrase 1 to Kinact for human recombinant carbonic anhydrase 5A | Homo sapiens | 27 | ALA1157705 | assay format | Scientific Literature | |
17. | ALA1068065 | B | Selectivity ratio of Kinact for human recombinant carbonic anhydrase 2 to Kinact for human recombinant carbonic anhydrase 5A | Homo sapiens | 26 | ALA1157705 | assay format | Scientific Literature | |
18. | ALA1068066 | B | Selectivity ratio of Kinact for human recombinant carbonic anhydrase 1 to Kinact for human recombinant carbonic anhydrase 5B | Homo sapiens | 26 | ALA1157705 | assay format | Scientific Literature | |
19. | ALA1068067 | B | Selectivity ratio of Kinact for human recombinant carbonic anhydrase 2 to Kinact for human recombinant carbonic anhydrase 5B | Homo sapiens | 26 | ALA1157705 | assay format | Scientific Literature | |
20. | ALA1614281 | F | PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Thyroid Stimulating Hormone Receptor: Activators of Intracellular cAMP Concentrations in Parental HEK 293. (Class of assay: confirmatory) | Homo sapiens | 12,194 | ALA1201862 | assay format | PubChem BioAssays |