| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA1059840 | F | Antagonist activity at human EP3 receptor expressed in cells assessed as mobilization of intracellular calcium by FLIPR assay | Homo sapiens | 24 | ALA1153033 | cell-based format | Scientific Literature | |
| 2. | ALA1059841 | B | Inhibition of human EP1 receptor by radioligand binding assay | Homo sapiens | 1 | ALA1153033 | single protein format | Scientific Literature | |
| 3. | ALA1060738 | B | Inhibition of human EP2 receptor by radioligand binding assay | Homo sapiens | 1 | ALA1153033 | single protein format | Scientific Literature | |
| 4. | ALA1060739 | B | Inhibition of human EP4 receptor by radioligand binding assay | Homo sapiens | 1 | ALA1153033 | single protein format | Scientific Literature | |
| 5. | ALA1060740 | B | Inhibition of human TP receptor by radioligand binding assay | Homo sapiens | 1 | ALA1153033 | single protein format | Scientific Literature | |
| 6. | ALA1060741 | B | Inhibition of human DP receptor | Homo sapiens | 2 | ALA1153033 | single protein format | Scientific Literature | |
| 7. | ALA1060742 | B | Displacement of [3H]PGF2a from human recombinant FP receptor expressed in HEK293 cells by scintillation counting | Homo sapiens | 1 | ALA1153033 | cell-based format | Scientific Literature | |
| 8. | ALA1060743 | B | Inhibition of COX1 in human whole blood by radioimmunoassay | Homo sapiens | 1 | ALA1153033 | tissue-based format | Scientific Literature | |
| 9. | ALA1060744 | B | Inhibition of COX2 in human whole blood by radioimmunoassay | Homo sapiens | 1 | ALA1153033 | tissue-based format | Scientific Literature | |
| 10. | ALA1060745 | B | Inhibition of rat EP3 receptor | Rattus norvegicus | 1 | ALA1153033 | single protein format | Scientific Literature | |
| 11. | ALA1060746 | B | Inhibition of dog EP3 receptor | Canis lupus familiaris | 1 | ALA1153033 | assay format | Scientific Literature | |
| 12. | ALA1060747 | F | Agonist activity at human EP3 receptor | Homo sapiens | 1 | ALA1153033 | assay format | Scientific Literature | |
| 13. | ALA1060757 | A | Half life in Sprague-Dawley rat at 2 mg/kg, po and 1 mg/kg, iv | Rattus norvegicus | 11 | ALA1153033 | organism-based format | Scientific Literature | |
| 14. | ALA1060758 | A | Clearance in Sprague-Dawley rat at 2 mg/kg, po and 1 mg/kg, iv | Rattus norvegicus | 11 | ALA1153033 | organism-based format | Scientific Literature | |
| 15. | ALA1060759 | A | Oral bioavailability in Sprague-Dawley rat at 2 mg/kg | Rattus norvegicus | 11 | ALA1153033 | organism-based format | Scientific Literature | |
| 16. | ALA3802311 | B | Displacement of [3H]PGE2 from human recombinant EP3 receptor expressed in human Chem1 cell membrane by scintillation proximity assay | Homo sapiens | 15 | ALA3797093 | cell-based format | Scientific Literature | |
| 17. | ALA3802312 | F | Antagonist activity at human recombinant EP3 receptor expressed in CHOK1 cells assessed as inhibition of sulprostone-induced decrease in cAMP level preincubated with compound followed by sulprostone addition by HTRF assay | Homo sapiens | 9 | ALA3797093 | cell-based format | Scientific Literature | |
| 18. | ALA3802313 | A | Apparent intrinsic clearance in human liver microsomes in presence of NADPH | Homo sapiens | 15 | ALA3797093 | tissue-based format | Scientific Literature | |
| 19. | ALA3802315 | A | Intrinsic clearance in human hepatocytes | Homo sapiens | 1 | ALA3797093 | cell-based format | Scientific Literature | |
| 20. | ALA3802316 | B | Displacement of [3H]PGE2 from human recombinant EP1 receptor expressed in human Chem1 cell membrane by scintillation proximity assay | Homo sapiens | 2 | ALA3797093 | cell-based format | Scientific Literature |
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