| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA1029353 | F | Antiproliferative activity against human PC3 cells at 4 uM after 48 hrs by MTT assay | Homo sapiens | 9 | ALA1158389 | cell-based format | Scientific Literature | |
| 2. | ALA1029354 | F | Antiproliferative activity against human SKOV3 cells at 4 uM after 48 hrs by MTT assay | Homo sapiens | 9 | ALA1158389 | cell-based format | Scientific Literature | |
| 3. | ALA1029355 | F | Antiproliferative activity against human A549 cells at 4 uM after 72 hrs by MTT assay | Homo sapiens | 9 | ALA1158389 | cell-based format | Scientific Literature | |
| 4. | ALA1029356 | F | Antiproliferative activity against human MIAPaCa2 cells at 4 uM after 48 hrs by MTT assay | Homo sapiens | 9 | ALA1158389 | cell-based format | Scientific Literature | |
| 5. | ALA1029357 | F | Antiproliferative activity against human BxPC3 cells at 4 uM after 48 hrs by MTT assay | Homo sapiens | 9 | ALA1158389 | cell-based format | Scientific Literature | |
| 6. | ALA1029358 | F | Antiproliferative activity against human T47D cells at 4 uM after 48 hrs by MTT assay | Homo sapiens | 9 | ALA1158389 | cell-based format | Scientific Literature | |
| 7. | ALA1029359 | F | Antiproliferative activity against human MDA-MB-468 cells at 4 uM after 48 hrs by MTT assay | Homo sapiens | 9 | ALA1158389 | cell-based format | Scientific Literature | |
| 8. | ALA1029365 | B | Transactivation of Gal4-LBD fused human RARalpha (156 to 454) transfected in african green monkey CV1 cells assessed as luciferase activity at 2 uM after 6 hrs by Dual-light chemiluminescent assay | Homo sapiens | 8 | ALA1158389 | cell-based format | Scientific Literature | |
| 9. | ALA1029366 | B | Transactivation of Gal4-LBD fused human RARbeta (169 to 448) transfected in african green monkey CV1 cells assessed as luciferase activity at 2 uM after 6 hrs by Dual-light chemiluminescent assay | Homo sapiens | 8 | ALA1158389 | cell-based format | Scientific Literature | |
| 10. | ALA1029367 | B | Transactivation of Gal4-LBD fused human RARgamma (178 to 454) transfected in african green monkey CV1 cells assessed as luciferase activity at 2 uM after 20 hrs by Dual-light chemiluminescent assay | Homo sapiens | 8 | ALA1158389 | cell-based format | Scientific Literature | |
| 11. | ALA1029368 | B | Inhibition of transactivation activity of Gal4-LBD fused human RARalpha (156 to 454) transfected in atRA-stimulated african green monkey CV1 cells at 4 uM after 6 hrs by Dual-light chemiluminescent assay | Homo sapiens | 4 | ALA1158389 | cell-based format | Scientific Literature | |
| 12. | ALA1029369 | B | Inhibition of transactivation activity of Gal4-LBD fused human RARalpha (156 to 454) transfected in atRA-stimulated african green monkey CV1 cells at 0.2 uM after 6 hrs by Dual-light chemiluminescent assay | Homo sapiens | 7 | ALA1158389 | cell-based format | Scientific Literature | |
| 13. | ALA1029370 | B | Inhibition of transactivation activity of Gal4-LBD fused human RARbeta (169 to 448) transfected in atRA-stimulated african green monkey CV1 cells at 4 uM after 6 hrs by Dual-light chemiluminescent assay | Homo sapiens | 7 | ALA1158389 | cell-based format | Scientific Literature | |
| 14. | ALA1029371 | B | Transactivation of Gal4-LBD fused mouse RXRalpha (218 to 467) transfected in african green monkey CV1 cells assessed as luciferase activity at 2 uM after 6 hrs by Dual-light chemiluminescent assay | Mus musculus | 5 | ALA1158389 | cell-based format | Scientific Literature | |
| 15. | ALA1029373 | B | Transactivation of Gal4-LBD fused mouse RXRalpha (218 to 467) transfected in african green monkey CV1 cells assessed as luciferase activity at after 6 hrs by Dual-light chemiluminescent assay | Mus musculus | 6 | ALA1158389 | cell-based format | Scientific Literature | |
| 16. | ALA1029374 | B | Inhibition of transactivation activity of Gal4-LBD fused human RARgamma (178 to 454) transfected in atRA-stimulated african green monkey CV1 cells at 4 uM after 6 hrs by Dual-light chemiluminescent assay | Homo sapiens | 7 | ALA1158389 | cell-based format | Scientific Literature | |
| 17. | ALA1031900 | F | Antiproliferative activity against human Jurkat T cells at 2 uM after 48 hrs by MTT assay | Homo sapiens | 2 | ALA1158389 | cell-based format | Scientific Literature | |
| 18. | ALA3118427 | B | Agonist activity at recombinant GST-tagged RXRalpha LBD (unknown origin) assessed as induction of biotinylated SRC-1-676-700 coactivator recruitment after 4 hrs by TR-FRET assay | Homo sapiens | 4 | ALA3112476 | single protein format | Scientific Literature | |
| 19. | ALA3118428 | B | Agonist activity at recombinant GST-tagged RXRalpha LBD (unknown origin) assessed as induction of fluorescein labeled D22 coactivator recruitment after 4 hrs by TR-FRET assay | Homo sapiens | 4 | ALA3112476 | single protein format | Scientific Literature | |
| 20. | ALA3118429 | B | Agonist activity at recombinant GST-tagged RXRalpha LBD (unknown origin) assessed as induction of biotinylated SRC-1-676-700 coactivator recruitment after 4 hrs by TR-FRET assay (Rvb = 148 +/- 7%) | Homo sapiens | 25 | ALA3112476 | single protein format | Scientific Literature |
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