| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA1057874 | F | Antagonist activity at human dopamine D3 receptor expressed in CHO cells by [35S]GTP-gamma-S-based scintillation spectrometry | Homo sapiens | 47 | cell-based format | Scientific Literature | ||
| 2. | ALA1057875 | F | Antagonist activity at human dopamine D2 receptor expressed in CHO cells by [35S]GTP-gamma-S-based scintillation spectrometry | Homo sapiens | 47 | cell-based format | Scientific Literature | ||
| 3. | ALA1057876 | B | Displacement of [3H]dofetilide from human ERG channel by scintillation proximity assay | Homo sapiens | 47 | single protein format | Scientific Literature | ||
| 4. | ALA1057877 | B | Selectivity ratio of pKi for human dopamine D3 receptor to pKi for human dopamine D2 receptor | Homo sapiens | 7 | assay format | Scientific Literature | ||
| 5. | ALA1057878 | A | Intrinsic clearance in human liver microsomes | Homo sapiens | 7 | microsome format | Scientific Literature | ||
| 6. | ALA1057879 | A | Intrinsic clearance in rat liver microsomes | Rattus norvegicus | 7 | microsome format | Scientific Literature | ||
| 7. | ALA1059862 | B | Binding affinity to human recombinant 5HT6 receptor expressed in CHO cells at 1 uM by radioligand binding assay | Homo sapiens | 1 | cell-based format | Scientific Literature | ||
| 8. | ALA1059863 | F | Antagonist activity at human D3 receptor expressed in CHO cells by [35S]GTPgammaS binding assay | Homo sapiens | 33 | cell-based format | Scientific Literature | ||
| 9. | ALA1059864 | F | Antagonist activity at human D2 receptor expressed in CHO cells by [35S]GTPgammaS binding assay | Homo sapiens | 33 | cell-based format | Scientific Literature | ||
| 10. | ALA1059865 | B | Displacement of [3H]dofetilide from human ERG channel by scintillation proximity assay | Homo sapiens | 33 | single protein format | Scientific Literature | ||
| 11. | ALA1059866 | B | Selectivity for human D3 receptor over human D2 receptor | Homo sapiens | 2 | assay format | Scientific Literature | ||
| 12. | ALA1059867 | B | Selectivity for human D3 receptor over human ERG | Homo sapiens | 2 | assay format | Scientific Literature | ||
| 13. | ALA1059868 | B | Binding affinity to human recombinant H1 receptor at 1 uM by radioligand binding assay | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 14. | ALA1059869 | B | Binding affinity to human recombinant muscarinic M1 receptor at 1 uM by radioligand binding assay | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 15. | ALA1059870 | B | Binding affinity to human recombinant muscarinic M2 receptor at 1 uM by radioligand binding assay | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 16. | ALA1059871 | B | Binding affinity to human recombinant muscarinic M3 receptor at 1 uM by radioligand binding assay | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 17. | ALA1059872 | B | Binding affinity to human recombinant muscarinic M4 receptor at 1 uM by radioligand binding assay | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 18. | ALA1059873 | B | Binding affinity to human recombinant muscarinic M5 receptor at 1 uM by radioligand binding assay | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 19. | ALA1059874 | B | Binding affinity to human recombinant 5HT1A receptor expressed in HEK293 cells at 1 uM by radioligand binding assay | Homo sapiens | 1 | cell-based format | Scientific Literature | ||
| 20. | ALA1059875 | B | Binding affinity to 5HT1B receptor in rat cortex at 1 uM by radioligand binding assay | Rattus norvegicus | 1 | tissue-based format | Scientific Literature |
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