# | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
---|---|---|---|---|---|---|---|---|---|
1. | ALA4359658 | Binding | Binding affinity to human C-terminal His8-tagged JAK2 pseudokinase (513 to 827 residues) expressed in baculovirus infected Hi-5 cells by intrinsic tryptophan fluorescence assay | Homo sapiens | 2 | ALA4354882 | cell-based format | Scientific Literature | |
2. | ALA4359660 | Binding | Binding affinity to wild type human C-terminal thrombin cleavage site-fused/ 6xHis-tagged JAK2 JH2 pseudokinase domain (536 to 812 residues) expressed in baculovirus infected sf9 insect cells measured for 1 hr in presence of fluorescein conjugate tracer by competitive fluorescence polarization assay | Homo sapiens | 15 | ALA4354882 | cell-based format | Scientific Literature | |
3. | ALA1060136 | Binding | Percentage IKK-beta activity remaining in the presence of 0.1uM inhibitor | Homo sapiens | 7 | ALA1150976 | single protein format | Scientific Literature | |
4. | ALA1060137 | Binding | Percentage JNK2 activity remaining in the presence of 0.1uM inhibitor | Homo sapiens | 7 | ALA1150976 | single protein format | Scientific Literature | |
5. | ALA1060139 | Binding | Percentage Lck activity remaining in the presence of 0.1uM inhibitor | Mus musculus | 7 | ALA1150976 | single protein format | Scientific Literature | |
6. | ALA1060140 | Binding | Percentage MAPKAPK2 activity remaining in the presence of 0.1uM inhibitor | Homo sapiens | 7 | ALA1150976 | single protein format | Scientific Literature | |
7. | ALA1060155 | Binding | Percentage PAK4 activity remaining in the presence of 0.1uM inhibitor | Homo sapiens | 7 | ALA1150976 | single protein format | Scientific Literature | |
8. | ALA1060156 | Binding | Percentage PKD1 activity remaining in the presence of 0.1uM inhibitor | Homo sapiens | 7 | ALA1150976 | single protein format | Scientific Literature | |
9. | ALA1060160 | Binding | Percentage Src activity remaining in the presence of 0.1uM inhibitor | Gallus gallus | 7 | ALA1150976 | single protein format | Scientific Literature | |
10. | ALA1060162 | Binding | Percentage SRPK1 activity remaining in the presence of 0.1uM inhibitor | Homo sapiens | 7 | ALA1150976 | single protein format | Scientific Literature | |
11. | ALA1061920 | Binding | Percentage CDK2-cyclinA activity remaining in the presence of 0.1uM inhibitor | Homo sapiens | 7 | ALA1150976 | protein complex format | Scientific Literature | |
12. | ALA1061947 | Binding | Percentage Aurora B activity remaining in the presence of 0.1uM inhibitor | Homo sapiens | 7 | ALA1150976 | single protein format | Scientific Literature | |
13. | ALA1061948 | Binding | Percentage Aurora C activity remaining in the presence of 0.1uM inhibitor | Homo sapiens | 7 | ALA1150976 | single protein format | Scientific Literature | |
14. | ALA1061953 | Binding | Percentage CK1delta activity remaining in the presence of 0.1uM inhibitor | Homo sapiens | 7 | ALA1150976 | single protein format | Scientific Literature | |
15. | ALA1061955 | Binding | Percentage DYRK2 activity remaining in the presence of 0.1uM inhibitor | Homo sapiens | 7 | ALA1150976 | single protein format | Scientific Literature | |
16. | ALA1061960 | Binding | Percentage ERK8 activity remaining in the presence of 0.1uM inhibitor | Homo sapiens | 7 | ALA1150976 | single protein format | Scientific Literature | |
17. | ALA1061961 | Binding | Percentage GSK3-beta activity remaining in the presence of 0.1uM inhibitor | Homo sapiens | 7 | ALA1150976 | single protein format | Scientific Literature | |
18. | ALA1061968 | Binding | Percentage JNK1 activity remaining in the presence of 0.1uM inhibitor | Homo sapiens | 7 | ALA1150976 | single protein format | Scientific Literature | |
19. | ALA1062768 | Binding | Percentage MST2 activity remaining in the presence of 0.1uM inhibitor | Homo sapiens | 7 | ALA1150976 | single protein format | Scientific Literature | |
20. | ALA1063718 | Binding | Percentage PAK5 activity remaining in the presence of 0.1uM inhibitor | Homo sapiens | 7 | ALA1150976 | single protein format | Scientific Literature |