| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA1046682 | B | Displacement of [125I]I-TAC from human CXCR3 expressed in CHO cells by scintillation proximity assay | Homo sapiens | 17 | ALA1154177 | cell-based format | Scientific Literature | |
| 2. | ALA1046683 | B | Displacement of [125I]I-TAC from mouse CXCR3 expressed in CHO cells by scintillation proximity assay | Mus musculus | 1 | ALA1154177 | cell-based format | Scientific Literature | |
| 3. | ALA1046684 | F | Antagonist activity at human CXCR3 expressed in L1.2 cells assessed as inhibition of I-TAC-induced Ca2+ mobilization by FLIPR assay | Homo sapiens | 17 | ALA1154177 | cell-based format | Scientific Literature | |
| 4. | ALA1046685 | F | Antagonist activity at mouse CXCR3 expressed in L1.2 cells assessed as inhibition of I-TAC-induced Ca2+ mobilization by FLIPR assay | Mus musculus | 1 | ALA1154177 | cell-based format | Scientific Literature | |
| 5. | ALA1046686 | F | Antagonist activity at human CXCR3 expressed in L1.2 cells assessed as inhibition of I-TAC-induced cell migration by flow cytometry | Homo sapiens | 1 | ALA1154177 | cell-based format | Scientific Literature | |
| 6. | ALA1046687 | A | Inhibition of CYP1A2 | 1 | ALA1154177 | single protein format | Scientific Literature | ||
| 7. | ALA1046688 | A | Inhibition of CYP2C9 | 1 | ALA1154177 | single protein format | Scientific Literature | ||
| 8. | ALA1046689 | A | Inhibition of CYP2C19 | 1 | ALA1154177 | single protein format | Scientific Literature | ||
| 9. | ALA1046690 | A | Inhibition of CYP2D6 | 1 | ALA1154177 | single protein format | Scientific Literature | ||
| 10. | ALA1046691 | A | Inhibition of CYP3A4 | 1 | ALA1154177 | single protein format | Scientific Literature | ||
| 11. | ALA1046692 | B | Inhibition of human ERG | Homo sapiens | 1 | ALA1154177 | single protein format | Scientific Literature | |
| 12. | ALA1046693 | P | Lipophilicity, log P of the compound | 1 | ALA1154177 | small-molecule physicochemical format | Scientific Literature | ||
| 13. | ALA1046694 | A | Intrinsic clearance in human | Homo sapiens | 1 | ALA1154177 | organism-based format | Scientific Literature | |
| 14. | ALA1046695 | A | Intrinsic clearance in rat | Rattus norvegicus | 1 | ALA1154177 | organism-based format | Scientific Literature | |
| 15. | ALA1046696 | P | Solubility in pH 1.0 buffer | 1 | ALA1154177 | small-molecule physicochemical format | Scientific Literature | ||
| 16. | ALA1046697 | P | Solubility in pH 6.8 buffer | 1 | ALA1154177 | small-molecule physicochemical format | Scientific Literature | ||
| 17. | ALA1046698 | A | Membrane permeability by PAMPA assay | 1 | ALA1154177 | assay format | Scientific Literature | ||
| 18. | ALA1046699 | A | Fraction unbound in human | Homo sapiens | 1 | ALA1154177 | organism-based format | Scientific Literature | |
| 19. | ALA1046700 | A | Fraction unbound in rat | Rattus norvegicus | 1 | ALA1154177 | organism-based format | Scientific Literature | |
| 20. | ALA1046701 | B | Inhibition of 5HT1A receptor | 2 | ALA1154177 | single protein format | Scientific Literature |
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