| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA1037630 | B | Binding affinity to human NK3 receptor | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 2. | ALA1037631 | B | Binding affinity to human NK2 receptor | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 3. | ALA1037632 | F | Agonist activity at human NK3 receptor expressed in cells assessed as accumulation of [3H]inositol phosphate | Homo sapiens | 1 | cell-based format | Scientific Literature | ||
| 4. | ALA1037633 | F | Agonist activity at guinea pig NK3 receptor expressed in cells assessed as accumulation of [3H]inositol phosphate | Cavia porcellus | 1 | cell-based format | Scientific Literature | ||
| 5. | ALA2215049 | B | Selectivity ratio of EC50 for human NK3 H316W mutant expressed in HEK293 cells to EC50 for wild type human NK3 receptor expressed in HEK293 cells | Homo sapiens | 1 | cell-based format | Scientific Literature | ||
| 6. | ALA2215050 | B | Selectivity ratio of EC50 for human NK3 Y247F mutant expressed in HEK293 cells to EC50 for wild type human NK3 receptor expressed in HEK293 cells | Homo sapiens | 1 | cell-based format | Scientific Literature | ||
| 7. | ALA2215516 | F | Agonist activity at human NK3 H316W mutant expressed in HEK293 cells assessed as [3H]IP accumulation after 45 mins | Homo sapiens | 1 | cell-based format | Scientific Literature | ||
| 8. | ALA2215517 | F | Agonist activity at human NK3 H316F mutant expressed in HEK293 cells assessed as [3H]IP accumulation after 45 mins | Homo sapiens | 1 | cell-based format | Scientific Literature | ||
| 9. | ALA2215518 | F | Agonist activity at human NK3 Y247W mutant expressed in HEK293 cells assessed as [3H]IP accumulation after 45 mins | Homo sapiens | 1 | cell-based format | Scientific Literature | ||
| 10. | ALA2215519 | F | Agonist activity at human NK3 Y247A mutant expressed in HEK293 cells assessed as [3H]IP accumulation after 45 mins | Homo sapiens | 1 | cell-based format | Scientific Literature | ||
| 11. | ALA2215520 | F | Agonist activity at human NK3 Y247F mutant expressed in HEK293 cells assessed as [3H]IP accumulation after 45 mins | Homo sapiens | 1 | cell-based format | Scientific Literature | ||
| 12. | ALA2210303 | F | Agonist activity at wild type human NK3 receptor expressed in HEK293 cells assessed as [3H]IP accumulation after 45 mins | Homo sapiens | 1 | cell-based format | Scientific Literature | ||
| 13. | ALA2210304 | B | Binding affinity at human NK1 receptor | Homo sapiens | 2 | single protein format | Scientific Literature | ||
| 14. | ALA2210305 | B | Binding affinity at human NK2 receptor | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 15. | ALA2350288 | B | Displacement of [125I]-NKA from NK2R (unknown origin) transfected in CHO cells at 10 uM by gamma counting analysis | Homo sapiens | 38 | cell-based format | Scientific Literature | ||
| 16. | ALA2350289 | B | Displacement of [125I]-BH-SP from NK1R (unknown origin) transfected in CHO cells at 10 uM by gamma counting analysis | Homo sapiens | 38 | cell-based format | Scientific Literature | ||
| 17. | ALA2350290 | F | Agonist activity at NK3R (unknown origin) transfected in CHO cells assessed as calcium influx at 10 mM | Homo sapiens | 38 | cell-based format | Scientific Literature | ||
| 18. | ALA2350291 | B | Displacement of ([125I]-His3, MePhe7)-NKB from NK3R (unknown origin) transfected in CHO cells by gamma counting analysis | Homo sapiens | 39 | cell-based format | Scientific Literature | ||
| 19. | ALA3372778 | B | Displacement of [125I]His3, MePhe7 from human NK3R expressed in CHO cell membranes by scintillation counting | Homo sapiens | 14 | cell-based format | Scientific Literature | ||
| 20. | ALA3373356 | F | Agonist activity at human NK3R expressed in CHO cells assessed as induction of Ca2+ influx by scintillation counting | Homo sapiens | 10 | cell-based format | Scientific Literature |
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