# | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
---|---|---|---|---|---|---|---|---|---|
1. | ALA1037224 | A | Binding affinity to human sex hormone binding globulin at 10 to 20 uCi/mL after 60 mins by instant thin layer chromatography | Homo sapiens | 2 | ALA1155242 | single protein format | Scientific Literature | |
2. | ALA1037226 | A | Binding affinity to rabbit sex hormone binding globulin at 10 to 20 uCi/mL after 60 mins by size-exclusion HPLC analysis | Oryctolagus cuniculus | 1 | ALA1155242 | single protein format | Scientific Literature | |
3. | ALA1037228 | A | Binding affinity to mouse serum albumin at 10 to 20 uCi/mL after 60 mins by size-exclusion HPLC analysis | Mus musculus | 3 | ALA1155242 | single protein format | Scientific Literature | |
4. | ALA1037230 | A | Stability in mouse serum assessed as intact compound remaining at 10 to 20 uCi/mL after 10 mins by size-exclusion HPLC analysis | Mus musculus | 1 | ALA1155242 | cell-free format | Scientific Literature | |
5. | ALA1037231 | A | Binding affinity to rabbit sex hormone binding globulin assessed as intact compound remaining at 10 to 20 uCi/mL after 60 mins by size-exclusion HPLC analysis | Oryctolagus cuniculus | 1 | ALA1155242 | single protein format | Scientific Literature | |
6. | ALA1037232 | A | Binding affinity to human sex hormone binding globulin assessed as intact compound remaining at 10 to 20 uCi/mL after 60 mins by instant thin layer chromatography | Homo sapiens | 1 | ALA1155242 | single protein format | Scientific Literature | |
7. | ALA1037239 | A | Stability in rabbit serum assessed as half life at 10 to 20 uCi/mL by size-exclusion HPLC analysis | Oryctolagus cuniculus | 1 | ALA1155242 | cell-free format | Scientific Literature | |
8. | ALA1037240 | A | Stability in human serum assessed as half life at 10 to 20 uCi/mL by size-exclusion HPLC analysis | Homo sapiens | 1 | ALA1155242 | cell-free format | Scientific Literature | |
9. | ALA1037241 | A | Stability in rabbit serum assessed as half life at 10 to 20 uCi/mL by reversed phase HPLC analysis | Oryctolagus cuniculus | 1 | ALA1155242 | cell-free format | Scientific Literature | |
10. | ALA1037242 | A | Stability in human serum assessed as half life at 10 to 20 uCi/mL by reversed phase HPLC analysis | Homo sapiens | 1 | ALA1155242 | cell-free format | Scientific Literature | |
11. | ALA1037243 | A | Binding affinity to rabbit sex hormone binding globulin at 10 to 20 uCi/mL after 60 mins by reversed phase HPLC analysis | Oryctolagus cuniculus | 1 | ALA1155242 | single protein format | Scientific Literature | |
12. | ALA1037245 | P | Chemical stability in phosphate buffer saline at 0.85 uCi after 1265 mins by HPLC analysis | 1 | ALA1155242 | small-molecule physicochemical format | Scientific Literature | ||
13. | ALA1037247 | P | Chemical stability in RPMI-1640 serum-free medium assessed as intact compound remaining at 12.2 uCi up to 6 hrs by HPLC analysis | 1 | ALA1155242 | small-molecule physicochemical format | Scientific Literature | ||
14. | ALA1037248 | P | Chemical stability in RPMI-1640 serum-free medium assessed as half life at 12.2 uCi by HPLC analysis | 1 | ALA1155242 | small-molecule physicochemical format | Scientific Literature | ||
15. | ALA1037249 | A | Stability in human OVCAR-3 cells expressing androgen receptor assessed as compound degradation at 0.1 uCi/mL up to 4 hrs by silica gel instant thin layer chromatography | Homo sapiens | 1 | ALA1155242 | cell-based format | Scientific Literature | |
16. | ALA1037250 | A | Stability in human OVCAR-3 cells expressing androgen receptor assessed as half life at 0.1 uCi/mL by silica gel instant thin layer chromatography | Homo sapiens | 1 | ALA1155242 | cell-based format | Scientific Literature | |
17. | ALA1037251 | A | Cellular uptake in single-cell suspension of nonproliferating human LNCAP cells expressing androgen receptor at 0.03 uCi/mL up to 2 hrs by gamma counting | Homo sapiens | 1 | ALA1155242 | cell-based format | Scientific Literature | |
18. | ALA1037252 | A | Cellular uptake in single-cell suspension of nonproliferating human LNCAP cells expressing androgen receptor assessed as increase in cellular retention at 0.37 uCi/mL after 5 to 16 hrs by gamma counting | Homo sapiens | 1 | ALA1155242 | cell-based format | Scientific Literature | |
19. | ALA1037253 | A | Cellular uptake in proliferating human LNCAP cells expressing androgen receptor after 24 hrs by gamma counting | Homo sapiens | 1 | ALA1155242 | cell-based format | Scientific Literature | |
20. | ALA1037259 | F | Cytotoxicity against human OVCAR-3 cells expressing androgen receptor assessed as cell survival at 0.01 to 5 uCi/mL after 24 hrs | Homo sapiens | 1 | ALA1155242 | cell-based format | Scientific Literature |