| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA1047183 | Binding | Inhibition of human PKCtheta by IMAP fluorescence polarization technology | Homo sapiens | 19 | ALA1156015 | single protein format | Scientific Literature | |
| 2. | ALA1047184 | Binding | Inhibition of PKCdelta by IMAP fluorescence polarization technology | 19 | ALA1156015 | single protein format | Scientific Literature | ||
| 3. | ALA1047185 | Binding | Ratio of IC50 for PKCdelta to IC50 for PKCdelta | 17 | ALA1156015 | assay format | Scientific Literature | ||
| 4. | ALA1047186 | ADME | Half life in rat liver microsomes | Rattus norvegicus | 1 | ALA1156015 | microsome format | Scientific Literature | |
| 5. | ALA1047187 | ADME | Half life in mouse liver microsomes | Mus musculus | 1 | ALA1156015 | microsome format | Scientific Literature | |
| 6. | ALA1047188 | ADME | Half life in human liver microsomes | Homo sapiens | 1 | ALA1156015 | microsome format | Scientific Literature | |
| 7. | ALA1047189 | ADME | Half life in dog liver microsomes | Canis lupus familiaris | 1 | ALA1156015 | microsome format | Scientific Literature | |
| 8. | ALA1047190 | ADME | Half life in monkey liver microsomes | Macaca mulatta | 1 | ALA1156015 | microsome format | Scientific Literature | |
| 9. | ALA1047191 | Binding | Inhibition of PKCtheta in C57BL/6 mouse T cells assessed as inhibition of anti-CD3 and anti-CD28-induced IL2 production after 20 to 24 hrs by ELISA | Mus musculus | 3 | ALA1156015 | cell-based format | Scientific Literature | |
| 10. | ALA1047192 | Functional | Inhibition of anti-CD3 and anti-CD28-induced IL2 production in PKCtheta knockout mouse after 20 to 24 hrs by ELISA | Mus musculus | 3 | ALA1156015 | organism-based format | Scientific Literature | |
| 11. | ALA1047193 | Binding | Inhibition of PKCbeta by IMAP fluorescence polarization technology | 1 | ALA1156015 | single protein format | Scientific Literature | ||
| 12. | ALA1047194 | Binding | Inhibition of PKCepsilon by IMAP fluorescence polarization technology | 1 | ALA1156015 | single protein format | Scientific Literature | ||
| 13. | ALA1047195 | Binding | Inhibition of PKCeta by IMAP fluorescence polarization technology | 1 | ALA1156015 | single protein format | Scientific Literature | ||
| 14. | ALA1047196 | Binding | Inhibition of PKCzeta by IMAP fluorescence polarization technology | 1 | ALA1156015 | single protein format | Scientific Literature | ||
| 15. | ALA1047197 | Binding | Inhibition of MK2 | 1 | ALA1156015 | single protein format | Scientific Literature | ||
| 16. | ALA1047198 | Binding | Inhibition of p38 | 1 | ALA1156015 | assay format | Scientific Literature | ||
| 17. | ALA1047199 | Binding | Inhibition of IKK | 1 | ALA1156015 | assay format | Scientific Literature | ||
| 18. | ALA1047200 | Binding | Inhibition of PDGFR | 1 | ALA1156015 | assay format | Scientific Literature | ||
| 19. | ALA1047201 | Binding | Inhibition of ROCK1 | 1 | ALA1156015 | single protein format | Scientific Literature | ||
| 20. | ALA1047202 | ADME | Membrane permeability by PAMPA | 1 | ALA1156015 | assay format | Scientific Literature |
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