| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA2157071 | B | Selectivity ratio of Ki for rat cloned dopamine D2L receptor to Ki for rat cloned dopamine D3 receptor | Rattus norvegicus | 24 | assay format | Scientific Literature | ||
| 2. | ALA2157072 | B | Displacement of [3H]spiroperidol from rat cloned dopamine D3 receptor expressed in HEK293 cells | Rattus norvegicus | 24 | cell-based format | Scientific Literature | ||
| 3. | ALA2157073 | B | Displacement of [3H]spiroperidol from rat cloned dopamine D2L receptor expressed in HEK293 cells | Rattus norvegicus | 24 | cell-based format | Scientific Literature | ||
| 4. | ALA2157074 | F | Agonist activity at human cloned dopamine D2 receptor expressed in CHO cells by [35S]GTPgammaS binding assay | Homo sapiens | 7 | cell-based format | Scientific Literature | ||
| 5. | ALA2157075 | F | Agonist activity at human cloned dopamine D2 receptor expressed in CHO cells by [35S]GTPgammaS binding assay relative to dopamine | Homo sapiens | 6 | cell-based format | Scientific Literature | ||
| 6. | ALA2157076 | F | Agonist activity at human cloned dopamine D3 receptor expressed in CHO cells by [35S]GTPgammaS binding assay | Homo sapiens | 7 | cell-based format | Scientific Literature | ||
| 7. | ALA2157077 | F | Agonist activity at human cloned dopamine D3 receptor expressed in CHO cells by [35S]GTPgammaS binding assay relative to dopamine | Homo sapiens | 6 | cell-based format | Scientific Literature | ||
| 8. | ALA2157078 | B | Selectivity ratio of EC50 for human cloned dopamine D2 receptor to EC50 for human cloned dopamine D3 receptor | Homo sapiens | 7 | assay format | Scientific Literature | ||
| 9. | ALA1050538 | B | Displacement of [3H]spiperone from human dopamine D3 receptor expressed in HEK293 cells | Homo sapiens | 17 | cell-based format | Scientific Literature | ||
| 10. | ALA1050539 | B | Displacement of [3H]spiperone from human dopamine D2L receptor expressed in HEK293 cells | Homo sapiens | 17 | cell-based format | Scientific Literature | ||
| 11. | ALA1050540 | B | Selectivity index, ratio of Ki for human dopamine D2L receptor to Ki for human dopamine D3 receptor | Homo sapiens | 17 | assay format | Scientific Literature | ||
| 12. | ALA1050541 | F | Agonist activity at human dopamine D2L receptor expressed in CHO cells assessed as stimulation of [35S]GTPgamma binding | Homo sapiens | 7 | cell-based format | Scientific Literature | ||
| 13. | ALA1050542 | F | Agonist activity at human dopamine D2L receptor expressed in CHO cells assessed as stimulation of [35S]GTPgamma binding relative to 1 mM dopamine | Homo sapiens | 6 | cell-based format | Scientific Literature | ||
| 14. | ALA1050543 | F | Agonist activity at human dopamine D3 receptor expressed in mouse AtT-20 cells assessed as stimulation of [35S]GTPgamma binding | Homo sapiens | 7 | cell-based format | Scientific Literature | ||
| 15. | ALA1050544 | F | Agonist activity at human dopamine D3 receptor expressed in mouse AtT-20 cells assessed as stimulation of [35S]GTPgamma binding relative to 100 uM dopamine | Homo sapiens | 6 | cell-based format | Scientific Literature | ||
| 16. | ALA1050545 | F | Selectivity index, ratio of EC50 for human dopamine D2L receptor to EC50 for human dopamine D3 receptor by [35S]GTPgamma binding assay | Homo sapiens | 7 | assay format | Scientific Literature | ||
| 17. | ALA1050546 | F | Antioxidant activity assessed as DPPH radical scavenging activity | 3 | assay format | Scientific Literature | |||
| 18. | ALA1050547 | F | Reversal of reserpine-induced hypolocomotion in Sprague-Dawley rat Parkinson's disease model at 10 umol/kg, sc measured after 6 hrs administered 18 hrs after reserpine challenge | Rattus norvegicus | 4 | organism-based format | Scientific Literature | ||
| 19. | ALA1050548 | F | Induction of rotational activity in 6-OHDA induced unilaterally lesioned Sprague-Dawley rat Parkinson's disease model assessed as duration of action at 10 umol/kg, sc | Rattus norvegicus | 3 | organism-based format | Scientific Literature | ||
| 20. | ALA1046239 | F | Induction of rotational activity in 6-OHDA induced unilaterally lesioned Sprague-Dawley rat Parkinson's disease model assessed as duration of action at 5 umol/kg, sc | Rattus norvegicus | 3 | organism-based format | Scientific Literature |
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