# | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
---|---|---|---|---|---|---|---|---|---|
1. | ALA1068015 | B | Inhibition of N type calcium channel alpha-1b/alpha-2-delta-1/beta-1b expressed in HEK293 cells at holding potential of -100 mV by whole-cell patch clamp method | 50 | cell-based format | Scientific Literature | |||
2. | ALA1068016 | B | Inhibition of L type calcium channel alpha-1c/alpha-2-delta-1/beta-1b expressed in HEK293 cells in presence of -100 mV holding potential by whole-cell patch clamp method | 13 | cell-based format | Scientific Literature | |||
3. | ALA1068017 | B | Inhibition of L-type calcium channel alpha-1c/alpha-2-delta-1/beta-1b expressed in HEK293 cells by FLIPR method | 23 | cell-based format | Scientific Literature | |||
4. | ALA3880754 | B | Antagonist activity at rat alpha1B N-type calcium channel expressed in HEK293 cells assessed as 0.067 Hz current frequency dependent channel blocking for 2 mins in presence of Ba2+ by whole-cell patch clamp assay | Rattus norvegicus | 33 | cell-based format | Patent Bioactivity Data | ||
5. | ALA3880755 | B | Antagonist activity at rat alpha1B N-type Ca2+ channel expressed in HEK293 cells assessed as 0.2 Hz current frequency dependent channel blocking for 2 mins in presence of Ba2+ by whole-cell patch clamp assay | Rattus norvegicus | 33 | cell-based format | Patent Bioactivity Data | ||
6. | ALA3880756 | B | Antagonist activity at rat brain alpha1B/alpha2b/beta1b N-type calcium channel expressed in HEK293 cells assessed as 0.1 Hz current frequency dependent channel blocking for 2 to 3 mins in presence of Ba2+ by whole-cell patch clamp assay | Rattus norvegicus | 6 | cell-based format | Patent Bioactivity Data | ||
7. | ALA3880757 | B | Antagonist activity at alpha1C/alpha2delta/beta1b L-type calcium channel (unknown origin) expressed in HEK293 cells assessed as 0.1 Hz current frequency dependent channel blocking for 2 to 3 mins in presence of Ba2+ by whole-cell patch clamp assay | Homo sapiens | 6 | cell-based format | Patent Bioactivity Data | ||
8. | ALA3880758 | B | Antagonist activity at alpha1A/alpha2delta/beta1b P/Q-type calcium channel (unknown origin) expressed in HEK293 cells assessed as 0.1 Hz current frequency dependent channel blocking for 2 to 3 mins in presence of Ba2+ by whole-cell patch clamp assay | Homo sapiens | 6 | cell-based format | Patent Bioactivity Data | ||
9. | ALA3880759 | B | Selectivity ratio of IC50 for alpha1A/alpha2delta/beta1b P/Q-type calcium channel (unknown origin) to IC50 for rat brain alpha1B/alpha2b/beta1b N-type calcium channel | 6 | assay format | Patent Bioactivity Data | |||
10. | ALA3880760 | B | Selectivity ratio of IC50 for alpha1C/alpha2delta/beta1b L-type calcium channel (unknown origin) to IC50 for rat brain alpha1B/alpha2b/beta1b N-type calcium channel | 6 | assay format | Patent Bioactivity Data |