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# Aladdin ID Assay Type Description Organism Compounds Reference BAO Format Source 1. ALA1104120 Binding Blocking of rat N-type calcium channel alpha-1B/alpha-2-delta-1/beta-1b activity expressed in HEK293 cells assessed as whole cell current by whole cell patch clamp assay Rattus norvegicus 25 ALA1154342 cell-based format Scientific Literature 2. ALA1116628 Binding Blocking of rat Voltage-dependent L-type calcium channel alpha1c/alpha2delta-1/beta1b activity expressed in HEK293 cells assessed as whole cell current by whole cell patch clamp assay Rattus norvegicus 10 ALA1154342 cell-based format Scientific Literature 3. ALA1116629 Binding Selectivity ratio of IC50 for rat Voltage-dependent L-type calcium channel to IC50 for rat N-type calcium channel Rattus norvegicus 10 ALA1154342 assay format Scientific Literature 4. ALA1116630 ADME Cmax in rat at 2 mg/kg, iv Rattus norvegicus 2 ALA1154342 organism-based format Scientific Literature 5. ALA1116631 ADME AUC (0 to 8 hrs) in rat at 2 mg/kg, iv Rattus norvegicus 2 ALA1154342 organism-based format Scientific Literature 6. ALA1116632 ADME AUC (0 to infinity) in rat at 2 mg/kg, iv Rattus norvegicus 2 ALA1154342 organism-based format Scientific Literature 7. ALA1116633 ADME Half life in rat at 2 mg/kg, iv Rattus norvegicus 2 ALA1154342 organism-based format Scientific Literature 8. ALA1116634 ADME Volume of distribution at steady state in rat at 2 mg/kg, iv Rattus norvegicus 2 ALA1154342 organism-based format Scientific Literature 9. ALA1116635 ADME Apparent oral clearance in rat at 2 mg/kg, iv Rattus norvegicus 2 ALA1154342 organism-based format Scientific Literature 10. ALA1116636 ADME Cmax in rat at 10 mg/kg, iv Rattus norvegicus 2 ALA1154342 organism-based format Scientific Literature 11. ALA1116637 ADME Tmax in rat at 10 mg/kg, iv Rattus norvegicus 2 ALA1154342 organism-based format Scientific Literature 12. ALA1116638 ADME AUC (0 to 8 hrs) in rat at 10 mg/kg, iv Rattus norvegicus 2 ALA1154342 organism-based format Scientific Literature 13. ALA1116639 ADME AUC (0 to infinity) in rat at 10 mg/kg, iv Rattus norvegicus 2 ALA1154342 organism-based format Scientific Literature 14. ALA1116640 ADME Half life in rat at 10 mg/kg, iv Rattus norvegicus 2 ALA1154342 organism-based format Scientific Literature 15. ALA1116641 ADME Apparent oral clearance in rat at 10 mg/kg, iv Rattus norvegicus 2 ALA1154342 organism-based format Scientific Literature 16. ALA1116642 ADME Oral bioavailability in rat at 10 mg/kg, iv Rattus norvegicus 2 ALA1154342 organism-based format Scientific Literature 17. ALA1116643 Functional Analgesic activity against phse 2A portion of rat formalin-induced inflammatory pain model assessed as flinches at 25 mg/kg, ip Rattus norvegicus 2 ALA1154342 organism-based format Scientific Literature 18. ALA1116644 Binding Inhibition of human ERG current at 1 uM Homo sapiens 2 ALA1154342 single protein format Scientific Literature