| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA1111355 | B | Displacement of [3H]Flumazenil from cloned human GABA alpha-5-beta-3-gamma-2 receptor expressed in HEK293 cells | Homo sapiens | 38 | ALA1154288 | cell-based format | Scientific Literature | |
| 2. | ALA1111359 | F | Inverse agonist activity at rat GABA alpha-5-beta-3-gamma-2 receptor expressed in HEK293 cells by electrophysiology assay relative to GABA | Rattus norvegicus | 31 | ALA1154288 | cell-based format | Scientific Literature | |
| 3. | ALA1111365 | B | Displacement of [3H]Flumazenil from cloned human GABA alpha-1-beta-3-gamma-2 receptor expressed in HEK293 cells | Homo sapiens | 6 | ALA1154288 | cell-based format | Scientific Literature | |
| 4. | ALA1111366 | B | Displacement of [3H]Flumazenil from cloned human GABA alpha-2-beta-3-gamma-2 receptor expressed in HEK293 cells | Homo sapiens | 6 | ALA1154288 | cell-based format | Scientific Literature | |
| 5. | ALA1111367 | B | Displacement of [3H]Flumazenil from cloned human GABA alpha-3-beta-3-gamma-2 receptor expressed in HEK293 cells | Homo sapiens | 6 | ALA1154288 | cell-based format | Scientific Literature | |
| 6. | ALA1111368 | F | Inverse agonist activity at rat GABA alpha-1-beta-3-gamma-2 receptor expressed in HEK293 cells by electrophysiology assay relative to GABA | Rattus norvegicus | 6 | ALA1154288 | cell-based format | Scientific Literature | |
| 7. | ALA1111369 | F | Inverse agonist activity at rat GABA alpha-2-beta-3-gamma-2 receptor expressed in HEK293 cells by electrophysiology assay relative to GABA | Rattus norvegicus | 6 | ALA1154288 | cell-based format | Scientific Literature | |
| 8. | ALA1111370 | F | Inverse agonist activity at rat GABA alpha-3-beta-3-gamma-2 receptor expressed in HEK293 cells by electrophysiology assay relative to GABA | Rattus norvegicus | 6 | ALA1154288 | cell-based format | Scientific Literature | |
| 9. | ALA1111371 | P | Solubility by lypophlisation solubility assay | 6 | ALA1154288 | small-molecule physicochemical format | Scientific Literature | ||
| 10. | ALA1111372 | P | Lipophilicity, log D at pH 7.4 | 6 | ALA1154288 | small-molecule physicochemical format | Scientific Literature | ||
| 11. | ALA1111373 | A | Permeability by PAMPA | 6 | ALA1154288 | assay format | Scientific Literature | ||
| 12. | ALA1111374 | A | Clearance in rat microsomes | Rattus norvegicus | 6 | ALA1154288 | microsome format | Scientific Literature | |
| 13. | ALA1111375 | A | Half life in rat | Rattus norvegicus | 6 | ALA1154288 | organism-based format | Scientific Literature | |
| 14. | ALA1111376 | A | Clearance in rat | Rattus norvegicus | 6 | ALA1154288 | organism-based format | Scientific Literature | |
| 15. | ALA1111377 | A | Volume of distribution at steady state in rat | Rattus norvegicus | 6 | ALA1154288 | organism-based format | Scientific Literature | |
| 16. | ALA1111378 | A | Oral bioavailability in rat | Rattus norvegicus | 6 | ALA1154288 | organism-based format | Scientific Literature | |
| 17. | ALA1111379 | A | Ratio of drug level in brain to plasma in rat | Rattus norvegicus | 6 | ALA1154288 | cell-free format | Scientific Literature | |
| 18. | ALA1111385 | A | Clearance in human microsomes | Homo sapiens | 6 | ALA1154288 | microsome format | Scientific Literature |
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