| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA1115172 | Binding | Binding affinity to 5HT2C receptor | 14 | ALA1156305 | single protein format | Scientific Literature | ||
| 2. | ALA1115173 | Binding | Binding affinity to 5HT2B receptor | 14 | ALA1156305 | single protein format | Scientific Literature | ||
| 3. | ALA1115174 | Binding | Selectivity ratio of Ki for 5HT2B receptor to Ki for 5HT2C receptor | 2 | ALA1156305 | assay format | Scientific Literature | ||
| 4. | ALA1115175 | Functional | Agonist activity at 5HT2C receptor | 8 | ALA1156305 | assay format | Scientific Literature | ||
| 5. | ALA1109735 | Functional | Agonist activity at 5HT2C receptor relative to control | 8 | ALA1156305 | assay format | Scientific Literature | ||
| 6. | ALA1109736 | Binding | Binding affinity to 5HT2A receptor | 4 | ALA1156305 | single protein format | Scientific Literature | ||
| 7. | ALA1109737 | Functional | Agonist activity at 5HT2B receptor | 4 | ALA1156305 | assay format | Scientific Literature | ||
| 8. | ALA1109739 | Functional | Agonist activity at 5HT2A receptor | 4 | ALA1156305 | assay format | Scientific Literature | ||
| 9. | ALA1109740 | Functional | Agonist activity at 5HT2A receptor relative to control | 4 | ALA1156305 | assay format | Scientific Literature | ||
| 10. | ALA1109741 | Functional | Ex vivo agonist activity at 5HT2B receptor in rat stomach fundus | Rattus norvegicus | 1 | ALA1156305 | organism-based format | Scientific Literature | |
| 11. | ALA1109742 | Binding | Activity at MAPK in monkey heart valve intestinal cells | Macaca mulatta | 1 | ALA1156305 | assay format | Scientific Literature | |
| 12. | ALA1109743 | Functional | Effect on 5HT2A receptor-mediated head twitches in rat | Rattus norvegicus | 1 | ALA1156305 | organism-based format | Scientific Literature | |
| 13. | ALA1109744 | Functional | Inhibition of spontaneous nocturnal food intake in po dosed Sprague-Dawley rat measured up to 840 mins | Rattus norvegicus | 1 | ALA1156305 | organism-based format | Scientific Literature | |
| 14. | ALA1109745 | Functional | Inhibition of spontaneous nocturnal food intake in po dosed Sprague-Dawley rat measured up to 25 hrs | Rattus norvegicus | 1 | ALA1156305 | organism-based format | Scientific Literature | |
| 15. | ALA1109746 | ADME | Fraction unbound in Sprague-Dawley rat plasma | Rattus norvegicus | 1 | ALA1156305 | cell-free format | Scientific Literature | |
| 16. | ALA1109747 | ADME | Ratio of drug level in RBC to plasma in Sprague-Dawley rat | Rattus norvegicus | 1 | ALA1156305 | assay format | Scientific Literature | |
| 17. | ALA1109748 | ADME | Ratio of total drug level in brain to plasma in Sprague-Dawley rat | Rattus norvegicus | 1 | ALA1156305 | cell-free format | Scientific Literature | |
| 18. | ALA1109749 | ADME | Ratio of free drug level in brain to plasma in Sprague-Dawley rat | Rattus norvegicus | 1 | ALA1156305 | cell-free format | Scientific Literature | |
| 19. | ALA1109750 | ADME | Bioavailability in rat | Rattus norvegicus | 1 | ALA1156305 | organism-based format | Scientific Literature | |
| 20. | ALA1109751 | ADME | Bioavailability in dog | Canis lupus familiaris | 1 | ALA1156305 | organism-based format | Scientific Literature |
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