| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA1105419 | ADME | Drug level in rat plasma at 50 mg/kg, po after 1 hr | Rattus norvegicus | 1 | ALA1156946 | organism-based format | Scientific Literature | |
| 2. | ALA1105420 | ADME | Drug level in rat brain at 50 mg/kg, po after 1 hr | Rattus norvegicus | 1 | ALA1156946 | organism-based format | Scientific Literature | |
| 3. | ALA1105421 | ADME | Ratio of drug level in rat brain to plasma at 50 mg/kg, po after 1 hr | Rattus norvegicus | 1 | ALA1156946 | organism-based format | Scientific Literature | |
| 4. | ALA1105422 | ADME | Drug level in mouse plasma at 50 mg/kg, po after 1 hr | Mus musculus | 1 | ALA1156946 | organism-based format | Scientific Literature | |
| 5. | ALA1105423 | ADME | Drug level in mouse brain at 50 mg/kg, po after 1 hr | Mus musculus | 1 | ALA1156946 | organism-based format | Scientific Literature | |
| 6. | ALA1105424 | ADME | Ratio of drug level in mouse brain to plasma at 50 mg/kg, po after 1 hr | Mus musculus | 1 | ALA1156946 | organism-based format | Scientific Literature | |
| 7. | ALA1105425 | Functional | Antiobesity activity in po dosed diet-induced obese mouse assessed as reduction in food intake after 14 days | Mus musculus | 1 | ALA1156946 | organism-based format | Scientific Literature | |
| 8. | ALA1105426 | Functional | Antiobesity activity in po dosed diet-induced obese mouse assessed as reduction in body weight after 14 days | Mus musculus | 1 | ALA1156946 | organism-based format | Scientific Literature | |
| 9. | ALA1116182 | Binding | Displacement of [125I]D-Tyr6-betaAla11-Phe13-Nle14-bombesin from human BRS-3 expressed in NFAT-CHO cells after 2 hrs by scintillation counting | Homo sapiens | 22 | ALA1156946 | cell-based format | Scientific Literature | |
| 10. | ALA1116183 | Functional | Agonist activity at human BRS-3 expressed in HEK293 cells coexpressing AEQ over 10 mins by aequorin bioluminescence assay | Homo sapiens | 22 | ALA1156946 | cell-based format | Scientific Literature | |
| 11. | ALA1116184 | Functional | Agonist activity at human BRS-3 expressed in HEK293 cells coexpressing AEQ over 10 mins by aequorin bioluminescence assay relative to D-Tyr6-betaAla11-Phe13-Nle14-bombesin | Homo sapiens | 22 | ALA1156946 | cell-based format | Scientific Literature | |
| 12. | ALA1116185 | Functional | Agonist activity at mouse BRS-3 expressed in HEK293 cells coexpressing AEQ over 10 mins by aequorin bioluminescence assay | Mus musculus | 22 | ALA1156946 | cell-based format | Scientific Literature | |
| 13. | ALA1116186 | Functional | Agonist activity at mouse BRS-3 expressed in HEK293 cells coexpressing AEQ over 10 mins by aequorin bioluminescence assay relative to D-Tyr6-betaAla11-Phe13-Nle14-bombesin | Mus musculus | 22 | ALA1156946 | cell-based format | Scientific Literature | |
| 14. | ALA1116187 | Binding | Displacement of [125I]D-Tyr6-betaAla11-Phe13-Nle14-bombesin from human NMB-R expressed in NFAT-CHO cells after 2 hrs by scintillation counting | Homo sapiens | 1 | ALA1156946 | cell-based format | Scientific Literature | |
| 15. | ALA1116188 | Binding | Displacement of [125I]D-Tyr6-betaAla11-Phe13-Nle14-bombesin from human GRP-R expressed in NFAT-CHO cells after 2 hrs by scintillation counting | Homo sapiens | 1 | ALA1156946 | cell-based format | Scientific Literature | |
| 16. | ALA1116189 | Binding | Displacement of [125I]D-Tyr6-betaAla11-Phe13-Nle14-bombesin from rat BRS-3 expressed in NFAT-CHO cells after 2 hrs by scintillation counting | Rattus norvegicus | 1 | ALA1156946 | cell-based format | Scientific Literature | |
| 17. | ALA1116190 | Binding | Displacement of [125I]D-Tyr6-betaAla11-Phe13-Nle14-bombesin from mouse BRS-3 expressed in NFAT-CHO cells after 2 hrs by scintillation counting | Mus musculus | 1 | ALA1156946 | cell-based format | Scientific Literature | |
| 18. | ALA1680282 | Functional | Agonist activity at human BRS-3 expressed in HEK293AEQ cells assessed as induction of intracellular calcium mobilization by aequorin bioluminescence assay | Homo sapiens | 8 | ALA1671827 | cell-based format | Scientific Literature | |
| 19. | ALA1680283 | Functional | Agonist activity at human BRS-3 expressed in HEK293AEQ cells assessed as induction of intracellular calcium mobilization by aequorin bioluminescence assay relative to dY peptide | Homo sapiens | 8 | ALA1671827 | cell-based format | Scientific Literature | |
| 20. | ALA1680284 | ADME | Half life in rat liver microsomes | Rattus norvegicus | 8 | ALA1671827 | microsome format | Scientific Literature |
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