| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA1116182 | Binding | Displacement of [125I]D-Tyr6-betaAla11-Phe13-Nle14-bombesin from human BRS-3 expressed in NFAT-CHO cells after 2 hrs by scintillation counting | Homo sapiens | 22 | ALA1156946 | cell-based format | Scientific Literature | |
| 2. | ALA1116183 | Functional | Agonist activity at human BRS-3 expressed in HEK293 cells coexpressing AEQ over 10 mins by aequorin bioluminescence assay | Homo sapiens | 22 | ALA1156946 | cell-based format | Scientific Literature | |
| 3. | ALA1116184 | Functional | Agonist activity at human BRS-3 expressed in HEK293 cells coexpressing AEQ over 10 mins by aequorin bioluminescence assay relative to D-Tyr6-betaAla11-Phe13-Nle14-bombesin | Homo sapiens | 22 | ALA1156946 | cell-based format | Scientific Literature | |
| 4. | ALA1116185 | Functional | Agonist activity at mouse BRS-3 expressed in HEK293 cells coexpressing AEQ over 10 mins by aequorin bioluminescence assay | Mus musculus | 22 | ALA1156946 | cell-based format | Scientific Literature | |
| 5. | ALA1116186 | Functional | Agonist activity at mouse BRS-3 expressed in HEK293 cells coexpressing AEQ over 10 mins by aequorin bioluminescence assay relative to D-Tyr6-betaAla11-Phe13-Nle14-bombesin | Mus musculus | 22 | ALA1156946 | cell-based format | Scientific Literature | |
| 6. | ALA1680281 | Binding | Displacement of [125I]-[D-Tyr6,beta-Ala11,Phe13,Nle14]-Bombesin (6-14) from human BRS-3 | Homo sapiens | 6 | ALA1671827 | single protein format | Scientific Literature | |
| 7. | ALA1680282 | Functional | Agonist activity at human BRS-3 expressed in HEK293AEQ cells assessed as induction of intracellular calcium mobilization by aequorin bioluminescence assay | Homo sapiens | 8 | ALA1671827 | cell-based format | Scientific Literature | |
| 8. | ALA1680283 | Functional | Agonist activity at human BRS-3 expressed in HEK293AEQ cells assessed as induction of intracellular calcium mobilization by aequorin bioluminescence assay relative to dY peptide | Homo sapiens | 8 | ALA1671827 | cell-based format | Scientific Literature | |
| 9. | ALA1680284 | ADME | Half life in rat liver microsomes | Rattus norvegicus | 8 | ALA1671827 | microsome format | Scientific Literature | |
| 10. | ALA1680290 | ADME | Plasma clearance in rat at 1 mg/kg, iv | Rattus norvegicus | 6 | ALA1671827 | organism-based format | Scientific Literature | |
| 11. | ALA1680291 | ADME | Faction unbound in human plasma at 1 uM | Homo sapiens | 6 | ALA1671827 | cell-free format | Scientific Literature | |
| 12. | ALA1680292 | ADME | Fraction unbound in rat plasma at 1 uM | Rattus norvegicus | 6 | ALA1671827 | cell-free format | Scientific Literature |
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