# | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
---|---|---|---|---|---|---|---|---|---|
1. | ALA638342 | A | Index of hydrophobicity (k') | 92 | ALA1123294 | assay format | Scientific Literature | ||
2. | ALA642476 | B | Evaluated for binding affinity against Adenosine A1 receptor | 17 | ALA1126162 | single protein format | Scientific Literature | ||
3. | ALA639501 | B | Molar potency ratio (MPR) against adenosine A2 receptor of canine coronary artery | Canis lupus familiaris | 85 | ALA1123294 | protein format | Scientific Literature | |
4. | ALA639504 | B | Acidic dissociation constant(pKa) against A2 adenosine receptor of coronary artery | Canis lupus familiaris | 34 | ALA1123294 | protein format | Scientific Literature | |
5. | ALA649129 | B | Displacement of [3H]-NECA from adenosine A2 receptor of rat striatal membrane | Rattus norvegicus | 14 | ALA1123754 | assay format | Scientific Literature | |
6. | ALA640604 | B | Displacement of [125I]ABA from adenosine A1 receptor of chick cerebellar membrane | Gallus gallus | 13 | ALA1123754 | assay format | Scientific Literature | |
7. | ALA636648 | B | Inhibition of binding of 1 nM N6-[3H]cyclohexyladenosine to adenosine A1 receptor on rat cerebral cortical membranes. | 19 | ALA1123049 | cell membrane format | Scientific Literature | ||
8. | ALA880535 | B | Relative affinities for adenosine A2 and A1 receptors | 14 | ALA1123754 | assay format | Scientific Literature | ||
9. | ALA1107960 | B | Displacement of [3H]CCPA from human adenosine A1 receptor expressed in CHO cells by scintillation counting | Homo sapiens | 7 | ALA1156209 | cell-based format | Scientific Literature | |
10. | ALA1107961 | B | Displacement of [3H]CCPA from human adenosine A1 receptor expressed in CHO cells by scintillation counting relative to control | Homo sapiens | 7 | ALA1156209 | cell-based format | Scientific Literature | |
11. | ALA1107962 | B | Displacement of [3H]DPCX from human adenosine A1 receptor expressed in CHO cells by scintillation counting | Homo sapiens | 10 | ALA1156209 | cell-based format | Scientific Literature | |
12. | ALA1107963 | B | Displacement of [3H]DPCX from human adenosine A1 receptor expressed in CHO cells by scintillation counting in presence of 10 uM allosteric modulator PD-81723 | Homo sapiens | 10 | ALA1156209 | cell-based format | Scientific Literature | |
13. | ALA1107964 | B | Selectivity ratio of Ki for human adenosine A1 receptor in presence of 10 uM allosteric modulator PD-81723 Ki for human adenosine A1 receptor | Homo sapiens | 10 | ALA1156209 | single protein format | Scientific Literature | |
14. | ALA1107965 | B | Displacement of [3H]DPCX from human adenosine A1 receptor expressed in CHO cells by scintillation counting relative to control | Homo sapiens | 10 | ALA1156209 | cell-based format | Scientific Literature | |
15. | ALA1107966 | F | Agonist activity at human adenosine A1 receptor expressed in CHO cells assessed as [35S]GTPgammaS binding by scintillation counting | Homo sapiens | 3 | ALA1156209 | cell-based format | Scientific Literature | |
16. | ALA1107967 | F | Agonist activity at human adenosine A1 receptor expressed in CHO cells assessed as [35S]GTPgammaS binding by scintillation counting in presence of 10 uM allosteric modulator PD-81723 | Homo sapiens | 3 | ALA1156209 | cell-based format | Scientific Literature | |
17. | ALA1107968 | F | Agonist activity at human adenosine A1 receptor expressed in CHO cells assessed as [35S]GTPgammaS binding by scintillation counting relative to control | Homo sapiens | 3 | ALA1156209 | cell-based format | Scientific Literature | |
18. | ALA1107969 | F | Agonist activity at human adenosine A1 receptor expressed in CHO cells assessed as [35S]GTPgammaS binding by scintillation counting in presence of 10 uM allosteric modulator PD-81723 relative to control | Homo sapiens | 3 | ALA1156209 | cell-based format | Scientific Literature | |
19. | ALA1107970 | B | Selectivity ratio of EC50 for human adenosine A1 receptor to EC50 for human adenosine A1 receptor in presence of 10 uM allosteric modulator PD-81723 | Homo sapiens | 3 | ALA1156209 | single protein format | Scientific Literature | |
20. | ALA1107971 | F | Agonist activity at human adenosine A1 receptor expressed in CHO cells assessed as stimulation of ERK1/2 phosphorylation | Homo sapiens | 3 | ALA1156209 | cell-based format | Scientific Literature |