| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA1104613 | Binding | Inhibition of human mTOR (1360-2549 amino acids) expressed in HEK293 cells | Homo sapiens | 49 | ALA1157009 | cell-based format | Scientific Literature | |
| 2. | ALA1104614 | Binding | Inhibition of PI3Kalpha by DELFIA assay | 49 | ALA1157009 | single protein format | Scientific Literature | ||
| 3. | ALA1104615 | Binding | Selectivity index, ratio of IC50 for PI3Kalpha to IC50 for human mTOR | 47 | ALA1157009 | assay format | Scientific Literature | ||
| 4. | ALA1104616 | Functional | Antiproliferative activity against human LNCAP cells after 3 days by MTS assay | Homo sapiens | 39 | ALA1157009 | cell-based format | Scientific Literature | |
| 5. | ALA1104617 | Binding | Inhibition of PI3Kgamma by DELFIA assay | 11 | ALA1157009 | single protein format | Scientific Literature | ||
| 6. | ALA1104618 | Binding | Inhibition of ATR by DELFIA assay | 11 | ALA1157009 | single protein format | Scientific Literature | ||
| 7. | ALA1104619 | ADME | Metabolic stability in mouse liver microsomes | Mus musculus | 15 | ALA1157009 | microsome format | Scientific Literature | |
| 8. | ALA1104621 | ADME | Inhibition of CYP2D6 at 3 uM | 15 | ALA1157009 | single protein format | Scientific Literature | ||
| 9. | ALA1104622 | ADME | Inhibition of CYP2C9 at 3 uM | 14 | ALA1157009 | single protein format | Scientific Literature | ||
| 10. | ALA1104623 | ADME | Inhibition of CYP3A4 at 3 uM | 15 | ALA1157009 | single protein format | Scientific Literature |
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