| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA1121100 | F | Agonist activity at histamine H2 receptor in spontaneously beating guinea pig atrium | Cavia porcellus | 11 | tissue-based format | Scientific Literature | ||
| 2. | ALA1121101 | F | Agonist activity at histamine H2 receptor in spontaneously beating guinea pig atrium assessed as increase in heart rate as relative to histamine | Cavia porcellus | 11 | tissue-based format | Scientific Literature | ||
| 3. | ALA1121102 | F | Agonist activity at GsalphaS-fused human histamine H2 receptor expressed in Sf9 cells by [35S]GTPgammaS binding assay relative to histamine | Homo sapiens | 11 | cell-based format | Scientific Literature | ||
| 4. | ALA1121103 | F | Agonist activity at GsalphaS-fused human histamine H2 receptor expressed in Sf9 cells by [35S]GTPgammaS binding assay | Homo sapiens | 11 | cell-based format | Scientific Literature | ||
| 5. | ALA1121104 | F | Agonist activity at GsalphaS-fused guinea pig histamine H2 receptor expressed in Sf9 cells by [35S]GTPgammaS binding assay relative to histamine | Cavia porcellus | 11 | cell-based format | Scientific Literature | ||
| 6. | ALA1121257 | F | Agonist activity at GsalphaS-fused guinea pig histamine H2 receptor expressed in Sf9 cells by [35S]GTPgammaS binding assay | Cavia porcellus | 11 | cell-based format | Scientific Literature | ||
| 7. | ALA1121258 | B | Selectivity ratio of EC50 for human histamine 5HT2 to EC50 for guinea pig 5HT2 receptor | 11 | assay format | Scientific Literature | |||
| 8. | ALA1121259 | B | Activity at human recombinant histamine H1 receptor expressed in Sf9 cells coexpressing RGS4 by steady-state GTPase activity assay | Homo sapiens | 11 | cell-based format | Scientific Literature | ||
| 9. | ALA1121261 | B | Activity at human recombinant histamine H3 receptor expressed in Sf9 cells coexpressing Galphai, Gbeta1gamma2 and RGS4 by steady-state GTPase activity assay | Homo sapiens | 11 | cell-based format | Scientific Literature | ||
| 10. | ALA1121263 | B | Activity at human recombinant GAIP-fused histamine H4 receptor expressed in Sf9 cells coexpressing Galphai, Gbeta1gamma2 by steady-state GTPase activity assay | Homo sapiens | 11 | cell-based format | Scientific Literature | ||
| 11. | ALA3225539 | B | Antagonist activity at guinea pig histamine H2 receptor assessed as inhibition of histamine-induced response after 30 mins | Cavia porcellus | 6 | single protein format | Scientific Literature | ||
| 12. | ALA3225542 | B | Antagonist activity at guinea pig ileum histamine H1 receptor assessed as inhibition of histamine-induced response after 10 to 15 mins | Cavia porcellus | 12 | tissue-based format | Scientific Literature | ||
| 13. | ALA3225911 | B | Agonist activity at guinea pig histamine H2 receptor assessed as potentiation of histamine-induced response after 30 mins | Cavia porcellus | 5 | single protein format | Scientific Literature |
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