| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA1109141 | Binding | Inhibition of GST-tagged PLK1 expressed in H5 insect cells assessed as [33P]gamma-ATP incorporation into substrate after 60 mins by gamma counting | 47 | ALA1157785 | cell-based format | Scientific Literature | ||
| 2. | ALA1109142 | Binding | Inhibition of Plk2 assessed as [33P]gamma-ATP incorporation into substrate after 60 mins by gamma counting | 25 | ALA1157785 | single protein format | Scientific Literature | ||
| 3. | ALA1109143 | Binding | Inhibition of Plk3 assessed as [33P]gamma-ATP incorporation into substrate after 60 mins by gamma counting | 25 | ALA1157785 | single protein format | Scientific Literature | ||
| 4. | ALA1109144 | Physicochemical | Solubility at pH 7 after 24 hrs by LC-MS/MS analysis | 25 | ALA1157785 | small-molecule physicochemical format | Scientific Literature | ||
| 5. | ALA1109145 | Binding | Inhibition of CDK2/Cyclin A assessed as [33P]gamma-ATP incorporation into substrate after 60 mins by gamma counting | 47 | ALA1157785 | protein complex format | Scientific Literature | ||
| 6. | ALA1109146 | Binding | Inhibition of Aurora A assessed as [33P]gamma-ATP incorporation into substrate after 60 mins by gamma counting | 47 | ALA1157785 | single protein format | Scientific Literature | ||
| 7. | ALA1109150 | Functional | Antiproliferative activity against human A2780 cells assessed as intracellular ATP level after 72 hrs by luminometry | Homo sapiens | 47 | ALA1157785 | cell-based format | Scientific Literature |
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