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| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source |
| 1. | ALA1103982 | Binding | Activity of glucokinase assessed as stimulatory concentration required to increase 1.5 fold enzymatic activity | | 58 | ALA1157747 | single protein format | Scientific Literature |
| 2. | ALA1103984 | Binding | Activation of glucokinase at 1 uM measured per mg of protein | | 2 | ALA1157747 | single protein format | Scientific Literature |
| 3. | ALA1103985 | Binding | Activation of glucokinase at 20 uM measured per mg of protein | | 2 | ALA1157747 | single protein format | Scientific Literature |
| 4. | ALA1103986 | Binding | Activation of glucokinase assessed as increase in Vmax at 1 uM relative to control | | 2 | ALA1157747 | single protein format | Scientific Literature |
| 5. | ALA1103987 | Binding | Activation of glucokinase at 20 uM relative to control | | 2 | ALA1157747 | single protein format | Scientific Literature |
| 6. | ALA1103988 | Binding | Activation of glucokinase assessed as increase in Km at 1 uM relative to control | | 2 | ALA1157747 | single protein format | Scientific Literature |
| 7. | ALA1103989 | Binding | Activation of glucokinase assessed as increase in Km at 20 uM relative to control | | 2 | ALA1157747 | single protein format | Scientific Literature |
| 8. | ALA1103990 | Binding | Activity of glucokinase up to 10 uM | | 2 | ALA1157747 | single protein format | Scientific Literature |
| 9. | ALA1103992 | Functional | Reduction of glucose-stimulated insulin secretion in C57BL/6J mouse isolated pancreatic islets cells after 3 to 4 days | Mus musculus | 2 | ALA1157747 | cell-based format | Scientific Literature |
| 10. | ALA1103993 | Functional | Reduction in glucose AUC in C57BL/6J mouse at 50 mg/kg, po pretreated 30 mins by oral glucose tolerance test relative to control | Mus musculus | 2 | ALA1157747 | organism-based format | Scientific Literature |
| 11. | ALA1103994 | ADME | Clearance in CD rat at 5 mg/kg, iv | Rattus norvegicus | 2 | ALA1157747 | organism-based format | Scientific Literature |
| 12. | ALA1103995 | ADME | Volume of distribution at steady state in CD rat at 5 mg/kg, iv | Rattus norvegicus | 2 | ALA1157747 | organism-based format | Scientific Literature |
| 13. | ALA1103996 | ADME | AUC (0 to infinity) in CD rat at 5 mg/kg, iv | Rattus norvegicus | 2 | ALA1157747 | organism-based format | Scientific Literature |
| 14. | ALA1103997 | ADME | AUC (0 to infinity) in CD rat at 10 mg/kg, po | Rattus norvegicus | 2 | ALA1157747 | organism-based format | Scientific Literature |
| 15. | ALA1103998 | ADME | AUC (0 to infinity) in CD rat at 30 mg/kg, po | Rattus norvegicus | 2 | ALA1157747 | organism-based format | Scientific Literature |
| 16. | ALA1103999 | ADME | Cmax in CD rat at 10 mg/kg, po | Rattus norvegicus | 2 | ALA1157747 | organism-based format | Scientific Literature |
| 17. | ALA1104000 | ADME | Cmax in CD rat at 30 mg/kg, po | Rattus norvegicus | 2 | ALA1157747 | organism-based format | Scientific Literature |
| 18. | ALA1104001 | ADME | Tmax in CD rat at 10 mg/kg, po | Rattus norvegicus | 2 | ALA1157747 | organism-based format | Scientific Literature |
| 19. | ALA1104002 | ADME | Tmax in CD rat at 30 mg/kg, po | Rattus norvegicus | 2 | ALA1157747 | organism-based format | Scientific Literature |
| 20. | ALA1104003 | ADME | Oral bioavailability in CD rat at 10 mg/kg | Rattus norvegicus | 2 | ALA1157747 | organism-based format | Scientific Literature |