# | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
---|---|---|---|---|---|---|---|---|---|
1. | ALA641504 | Binding | Binding affinity against AMPA receptor in rat brain membrane using [3H]-AMPA as radioligand | 22 | ALA1127329 | cell membrane format | Scientific Literature | ||
2. | ALA644192 | Binding | Binding affinity against AMPA receptor using [3H]- AMPA radioligand | 15 | ALA1130361 | protein complex format | Scientific Literature | ||
3. | ALA702871 | Binding | In vitro inhibition of [3H]KAIN binding to Ionotropic glutamate receptor kainate. | 20 | ALA1129553 | protein complex format | Scientific Literature | ||
4. | ALA702875 | Binding | Displacement of [3H]CNQX from Ionotropic glutamate receptor kainate/Ionotropic glutamate receptor AMPA in rat cortical membranes | Rattus norvegicus | 11 | ALA1127957 | cell membrane format | Scientific Literature | |
5. | ALA697170 | Binding | In vitro inhibition of [3H]AMPA binding to Ionotropic glutamate receptor AMPA. | 21 | ALA1129553 | protein complex format | Scientific Literature | ||
6. | ALA697794 | Binding | Inhibition of specific binding of [3H]AMPA to Ionotropic glutamate receptor AMPA in rat brain membranes | 8 | ALA1130171 | cell membrane format | Scientific Literature | ||
7. | ALA697800 | Binding | Tested for the inhibition of binding of [3H]AMPA radioligand to Ionotropic glutamate receptor AMPA to cortical membranes from rat brain | 7 | ALA1126991 | assay format | Scientific Literature | ||
8. | ALA697375 | Binding | Binding affinity for Ionotropic glutamate receptor AMPA was determined by the ability to displace [3H]AMPA in rat cortical membranes | 6 | ALA1127000 | cell membrane format | Scientific Literature | ||
9. | ALA701236 | Binding | In vitro inhibition of [3H]CNQX binding to Ionotropic glutamate receptor AMPA. | 20 | ALA1129553 | protein complex format | Scientific Literature | ||
10. | ALA696376 | Binding | Inhibition of specific binding of [3H]kainate to Ionotropic glutamate receptor kainate in rat brain membranes | 9 | ALA1130171 | cell membrane format | Scientific Literature | ||
11. | ALA696380 | Binding | Tested for the inhibition of binding of [3H]kainate radioligand to Ionotropic glutamate receptor kainate of cortical membranes from rat brain | 7 | ALA1126991 | assay format | Scientific Literature | ||
12. | ALA698700 | Binding | Binding affinity against kainate receptor in rat brain membrane using [3H]kainate as radioligand | 3 | ALA1127329 | cell membrane format | Scientific Literature | ||
13. | ALA862719 | Functional | Antagonism on GLUK5 containing kainate induced depolarization of isolated neonatal rat dorsal root C-fibers | Rattus norvegicus | 18 | ALA1141230 | assay format | Scientific Literature | |
14. | ALA862730 | Binding | Displacement of [3H]kainate from rat GLUK6 receptor expressed in HEK293 cells | Rattus norvegicus | 21 | ALA1141230 | cell-based format | Scientific Literature | |
15. | ALA861532 | Functional | Antagonist activity against GLUK5-containing kainate receptor by inhibition of kainate-induced depolarization of neonatal rat dorsal root fibers | 14 | ALA1146072 | assay format | Scientific Literature | ||
16. | ALA866869 | Functional | Antagonist activity against AMPA receptor expressed in motoneurones by inhibition of fDR-VRP in the neonatal rat spinal cord | Rattus norvegicus | 16 | ALA1146072 | assay format | Scientific Literature | |
17. | ALA865634 | Binding | Displacement of [3H]kainate from rat GLUK6 expressed in HEK293 cells | Rattus norvegicus | 15 | ALA1146072 | cell-based format | Scientific Literature | |
18. | ALA870672 | Functional | Antagonist activity against rat KA receptor assessed by inhibition of kainate-induced membrane current at 1 uM | Rattus norvegicus | 1 | ALA1146962 | assay format | Scientific Literature | |
19. | ALA904263 | Functional | Activity at native GLUK5 kainate receptor assessed as antagonism of kainite-induced depolarization of neonatal anaesthetised rat dorsal root fibres | Rattus norvegicus | 14 | ALA1142988 | assay format | Scientific Literature | |
20. | ALA1106352 | Functional | Antagonist activity at recombinant GluA1A2 receptor flip isoform expressed in Xenopus oocytes | 2 | ALA1157033 | cell-based format | Scientific Literature |