| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA1120617 | Binding | Displacement of [125I]cyanopindolol from human adrenergic beta-1 receptor expressed in CHOK1 cells | Homo sapiens | 34 | ALA1155476 | cell-based format | Scientific Literature | |
| 2. | ALA1120618 | Binding | Displacement of [125I]cyanopindolol from human adrenergic beta2 receptor expressed in CHOK1 cells | Homo sapiens | 34 | ALA1155476 | cell-based format | Scientific Literature | |
| 3. | ALA1120619 | Binding | Displacement of [125I]cyanopindolol from human adrenergic beta3 receptor expressed in CHOK1 cells | Homo sapiens | 34 | ALA1155476 | cell-based format | Scientific Literature | |
| 4. | ALA1120620 | Functional | Agonist activity at human adrenergic beta-1 receptor expressed in CHOK1 cells assessed as cAMP accumulation by HTRF assay | Homo sapiens | 2 | ALA1155476 | cell-based format | Scientific Literature | |
| 5. | ALA1120621 | Functional | Intrinsic activity at human adrenergic beta-1 receptor expressed in CHOK1 cells assessed as cAMP accumulation by HTRF assay relative to isoproterenol | Homo sapiens | 2 | ALA1155476 | cell-based format | Scientific Literature | |
| 6. | ALA1117707 | Functional | Antagonist activity at human adrenergic beta2 receptor expressed in CHOK1 cells assessed as inhibition of cAMP accumulation by HTRF assay | Homo sapiens | 2 | ALA1155476 | cell-based format | Scientific Literature | |
| 7. | ALA1117708 | Functional | Agonist activity at human adrenergic beta3 receptor expressed in CHOK1 cells assessed as cAMP accumulation by HTRF assay | Homo sapiens | 4 | ALA1155476 | cell-based format | Scientific Literature | |
| 8. | ALA1117709 | Functional | Intrinsic activity at human adrenergic beta3 receptor expressed in CHOK1 cells assessed as cAMP accumulation by HTRF assay relative to isoproterenol | Homo sapiens | 4 | ALA1155476 | cell-based format | Scientific Literature | |
| 9. | ALA1117711 | Physicochemical | Solubility at pH 4 | 1 | ALA1155476 | small-molecule physicochemical format | Scientific Literature | ||
| 10. | ALA1117712 | Physicochemical | Solubility at pH 6 | 1 | ALA1155476 | small-molecule physicochemical format | Scientific Literature | ||
| 11. | ALA1117713 | ADME | Permeability by PAMPA method | 1 | ALA1155476 | assay format | Scientific Literature | ||
| 12. | ALA1117714 | ADME | Cytotoxicity against human PBMC cells | Homo sapiens | 1 | ALA1155476 | cell-based format | Scientific Literature | |
| 13. | ALA1117715 | ADME | Cytotoxicity against human HepG2 cells | Homo sapiens | 1 | ALA1155476 | cell-based format | Scientific Literature | |
| 14. | ALA1117716 | ADME | Cmax in Wistar rat at 10 mg/kg, po | Rattus norvegicus | 1 | ALA1155476 | organism-based format | Scientific Literature | |
| 15. | ALA1117717 | ADME | Half life in Wistar rat at 10 mg/kg, po | Rattus norvegicus | 1 | ALA1155476 | organism-based format | Scientific Literature |
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