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| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source |
| 1. | ALA680747 | Binding | Selectivity for gardos channel; (Gardos channel vs 2000 nM for the cardiac IKs channel).) | | 1 | ALA1134478 | protein complex format | Scientific Literature |
| 2. | ALA948111 | Binding | Inhibition of Gardos channel in human RBC assessed as inhibition of ionomycin-stimulated [86Rb] efflux | Homo sapiens | 23 | ALA1141563 | single protein format | Scientific Literature |
| 3. | ALA948112 | ADME | Intrinsic clearance in rat liver microsome S9 fraction as % compound remaining after incubation | Rattus norvegicus | 15 | ALA1141563 | subcellular format | Scientific Literature |
| 4. | ALA948113 | Physicochemical | Solubility by shake-flask method | | 15 | ALA1141563 | small-molecule physicochemical format | Scientific Literature |
| 5. | ALA948114 | ADME | Bioavailability in Sprague-Dawley rat at 1 mg/kg, iv or 10 mg/kg, po | Rattus norvegicus | 2 | ALA1141563 | organism-based format | Scientific Literature |
| 6. | ALA948115 | ADME | Half life in Sprague-Dawley rat at 1 mg/kg, iv or 10 mg/kg, po | Rattus norvegicus | 2 | ALA1141563 | organism-based format | Scientific Literature |
| 7. | ALA948116 | ADME | Tmax in Sprague-Dawley rat at 1 mg/kg, iv or 10 mg/kg, po | Rattus norvegicus | 2 | ALA1141563 | organism-based format | Scientific Literature |
| 8. | ALA948117 | ADME | Cmax in Sprague-Dawley rat at 1 mg/kg, iv or 10 mg/kg, po | Rattus norvegicus | 2 | ALA1141563 | organism-based format | Scientific Literature |
| 9. | ALA948119 | ADME | Inhibition of CYP3A4 at 10 uM | | 5 | ALA1141563 | single protein format | Scientific Literature |
| 10. | ALA948121 | Functional | Effect on gardos channel activity in SAD1 mouse model assessed by measuring [86Rb]/L of cells at 20 mg/kg, po bid after 7 days | Mus musculus | 1 | ALA1141563 | organism-based format | Scientific Literature |
| 11. | ALA948122 | Functional | Effect on gardos channel activity in SAD1 mouse model assessed by measuring [86Rb]/L of cells at 20 mg/kg, po bid after 14 days | Mus musculus | 1 | ALA1141563 | organism-based format | Scientific Literature |
| 12. | ALA948123 | Functional | Effect on mean corpuscular hemoglobin concentration in SAD1 mouse model at 20 mg/kg, po bid after 7 days | Mus musculus | 1 | ALA1141563 | organism-based format | Scientific Literature |
| 13. | ALA948124 | Functional | Effect on mean corpuscular hemoglobin concentration in SAD1 mouse model at 20 mg/kg, po bid after 14 days | Mus musculus | 1 | ALA1141563 | organism-based format | Scientific Literature |
| 14. | ALA948125 | Functional | Effect on hematocrit levels in SAD1 mouse model at 20 mg/kg, po bid after 7 days | Mus musculus | 1 | ALA1141563 | organism-based format | Scientific Literature |
| 15. | ALA948126 | Functional | Effect on hematocrit levels in SAD1 mouse model at 20 mg/kg, po bid after 14 days | Mus musculus | 1 | ALA1141563 | organism-based format | Scientific Literature |
| 16. | ALA819394 | Binding | Inhibition of Iks current KvLQT1 potassium channel | | 1 | ALA1134478 | protein complex format | Scientific Literature |