| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA3772516 | B | Inhibition of human recombinant KLK4 expressed in Escherichia coli using Bachem I-1120 as substrate preincubated for 15 mins followed by substrate addition by microplate reader analysis | Homo sapiens | 11 | ALA3769401 | assay format | Scientific Literature | |
| 2. | ALA3772517 | B | Inhibition of human recombinant KLK2 expressed in Escherichia coli using Bachem I-1295 as substrate preincubated for 15 mins followed by substrate addition by microplate reader analysis | Homo sapiens | 11 | ALA3769401 | assay format | Scientific Literature | |
| 3. | ALA3772518 | B | Inhibition of human recombinant KLK1 expressed in Escherichia coli using Bachem I-1295 as substrate preincubated for 15 mins followed by substrate addition by microplate reader analysis | Homo sapiens | 11 | ALA3769401 | assay format | Scientific Literature | |
| 4. | ALA3772679 | B | Inhibition of human recombinant KLK8 expressed in Escherichia coli using Bachem I-1120 as substrate preincubated for 15 mins followed by substrate addition by microplate reader analysis | Homo sapiens | 11 | ALA3769401 | assay format | Scientific Literature | |
| 5. | ALA3772680 | B | Inhibition of recombinant uPA (unknown origin) using Biophen CS-61(44) as substrate | Homo sapiens | 11 | ALA3769401 | single protein format | Scientific Literature | |
| 6. | ALA3772681 | B | Inhibition of recombinant tPA (unknown origin) using Biophen CS-05(88) as substrate | Homo sapiens | 11 | ALA3769401 | single protein format | Scientific Literature | |
| 7. | ALA3772682 | B | Inhibition of human plasma thrombin using Biophen CS-21(66) as substrate preincubated for 15 mins followed by substrate addition by microplate reader analysis | Homo sapiens | 11 | ALA3769401 | cell-free format | Scientific Literature | |
| 8. | ALA3772683 | B | Inhibition of human plasma plasmin using Biophen CS-21(66) as substrate | Homo sapiens | 10 | ALA3769401 | cell-free format | Scientific Literature | |
| 9. | ALA3772684 | B | Inhibition of factor 10a (unknown origin) using Biophen CS-11(32) as substrate | Homo sapiens | 11 | ALA3769401 | single protein format | Scientific Literature | |
| 10. | ALA3772685 | B | Inhibition of Electrophorus electricus AChE using acetylthiocholine iodide as substrate by 5-5'-Dithiobis(2 nitrobenzoic acid)-based assay | Electrophorus electricus | 10 | ALA3769401 | single protein format | Scientific Literature | |
| 11. | ALA3772686 | B | Reversible inhibition of human recombinant KLK2 expressed in Escherichia coli using H-Pro-Phe-Arg-AMC as fluorogenic substrate at 100 times IC50 preincubated for 15 mins followed by 100 fold dilution measured for 1 hr | Homo sapiens | 3 | ALA3769401 | assay format | Scientific Literature | |
| 12. | ALA3772688 | B | Reversible inhibition of human recombinant KLK1 expressed in Escherichia coli using H-Pro-Phe-Arg-AMC as fluorogenic substrate at 100 times IC50 preincubated for 15 mins followed by 100 fold dilution measured for 1 hr | Homo sapiens | 1 | ALA3769401 | assay format | Scientific Literature | |
| 13. | ALA3772695 | B | Selectivity ratio of IC50 for human recombinant KLK2 to IC50 for human recombinant KLK4 | Homo sapiens | 1 | ALA3769401 | assay format | Scientific Literature | |
| 14. | ALA3772696 | B | Selectivity ratio of IC50 for human recombinant KLK1 to IC50 for human recombinant KLK4 | Homo sapiens | 1 | ALA3769401 | assay format | Scientific Literature | |
| 15. | ALA3772697 | B | Selectivity ratio of IC50 for human recombinant KLK8 to IC50 for human recombinant KLK4 | Homo sapiens | 1 | ALA3769401 | assay format | Scientific Literature | |
| 16. | ALA3772698 | B | Selectivity ratio of IC50 for recombinant uPA (unknown origin) to IC50 for human recombinant KLK4 | Homo sapiens | 1 | ALA3769401 | assay format | Scientific Literature | |
| 17. | ALA3772699 | B | Selectivity ratio of IC50 for recombinant tPA (unknown origin) to IC50 for human recombinant KLK4 | Homo sapiens | 1 | ALA3769401 | assay format | Scientific Literature | |
| 18. | ALA3772700 | B | Selectivity ratio of IC50 for human plasma thrombin to IC50 for human recombinant KLK4 | Homo sapiens | 1 | ALA3769401 | assay format | Scientific Literature | |
| 19. | ALA3772701 | B | Selectivity ratio of IC50 for human plasma plasmin to IC50 for human recombinant KLK4 | Homo sapiens | 1 | ALA3769401 | assay format | Scientific Literature | |
| 20. | ALA3772702 | B | Selectivity ratio of IC50 for factor 10a (unknown origin) to IC50 for human recombinant KLK4 | Homo sapiens | 1 | ALA3769401 | assay format | Scientific Literature |
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