| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA3105981 | B | Competitive inhibition of DYRK1A (unknown origin) using ATP | Homo sapiens | 2 | single protein format | Scientific Literature | ||
| 2. | ALA3599536 | B | Inhibition of Dyrk1A (unknown origin) | Homo sapiens | 2 | single protein format | Scientific Literature | ||
| 3. | ALA4266661 | B | Inhibition of human recombinant full length GST-tagged DYRK1A expressed in baculovirus expression system after 10 mins in presence of [gamma33P-ATP] by liquid scintillation counting analysis | Homo sapiens | 2 | assay format | Scientific Literature | ||
| 4. | ALA5096128 | F | In vitro activity on S. mansoni schistosomula at 50 uM | Schistosoma mansoni | 80 | organism-based format | Cardiff Schistosomiasis Dataset 2023 | ||
| 5. | ALA5096129 | F | In vitro activity on S. mansoni schistosomula at 10 uM | Schistosoma mansoni | 80 | organism-based format | Cardiff Schistosomiasis Dataset 2023 | ||
| 6. | ALA5251363 | B | Inhibition of recombinant human CDK5/p25 expressed in Sf9 insect cells incubated for 60 mins in presence of ATP and [gamma33-P] ATP by radiometric scintillation counter analysis | Homo sapiens | 56 | cell-based format | Scientific Literature | ||
| 7. | ALA5251364 | B | Inhibition of recombinant human CK1epsilon expressed in Sf9 insect cells incubated for 60 mins in presence of ATP and [gamma33-P] ATP by radiometric scintillation counter analysis | Homo sapiens | 56 | cell-based format | Scientific Literature | ||
| 8. | ALA5251365 | B | Inhibition of recombinant human CLK1 expressed in Sf9 insect cells incubated for 60 mins in presence of ATP and [gamma33-P] ATP by radiometric scintillation counter analysis | Homo sapiens | 56 | cell-based format | Scientific Literature | ||
| 9. | ALA5251366 | B | Inhibition of recombinant human CLK2 expressed in Sf9 insect cells incubated for 60 mins in presence of ATP and [gamma33-P] ATP by radiometric scintillation counter analysis | Homo sapiens | 56 | cell-based format | Scientific Literature | ||
| 10. | ALA5251367 | B | Inhibition of recombinant human CLK3 expressed in Sf9 insect cells incubated for 60 mins in presence of ATP and [gamma33-P] ATP by radiometric scintillation counter analysis | Homo sapiens | 56 | cell-based format | Scientific Literature | ||
| 11. | ALA5251368 | B | Inhibition of recombinant human CLK4 expressed in Sf9 insect cells incubated for 60 mins in presence of ATP and [gamma33-P] ATP by radiometric scintillation counter analysis | Homo sapiens | 56 | cell-based format | Scientific Literature | ||
| 12. | ALA5251369 | B | Inhibition of recombinant human DYRK1A expressed in Sf9 insect cells incubated for 60 mins in presence of ATP and [gamma33-P] ATP by radiometric scintillation counter analysis | Homo sapiens | 56 | cell-based format | Scientific Literature | ||
| 13. | ALA5251370 | B | Inhibition of recombinant human DYRK1B expressed in Sf9 insect cells incubated for 60 mins in presence of ATP and [gamma33-P] ATP by radiometric scintillation counter analysis | Homo sapiens | 56 | cell-based format | Scientific Literature | ||
| 14. | ALA5251371 | B | Inhibition of recombinant human DYRK2 expressed in Sf9 insect cells incubated for 60 mins in presence of ATP and [gamma33-P] ATP by radiometric scintillation counter analysis | Homo sapiens | 56 | cell-based format | Scientific Literature | ||
| 15. | ALA5251372 | B | Inhibition of recombinant human DYRK3 expressed in Sf9 insect cells incubated for 60 mins in presence of ATP and [gamma33-P] ATP by radiometric scintillation counter analysis | Homo sapiens | 56 | cell-based format | Scientific Literature | ||
| 16. | ALA5251373 | B | Inhibition of recombinant human DYRK4 expressed in Sf9 insect cells incubated for 60 mins in presence of ATP and [gamma33-P] ATP by radiometric scintillation counter analysis | Homo sapiens | 56 | cell-based format | Scientific Literature | ||
| 17. | ALA5251374 | B | Inhibition of recombinant human GSK-3beta expressed in Sf9 insect cells incubated for 60 mins in presence of ATP and [gamma33-P] ATP by radiometric scintillation counter analysis | Homo sapiens | 56 | cell-based format | Scientific Literature | ||
| 18. | ALA5251375 | B | Selectivity ratio of IC50 for recombinant human CLK1 expressed in Sf9 insect cells to IC50 for recombinant human DYRK1A expressed in Sf9 insect cells | Homo sapiens | 46 | cell-based format | Scientific Literature | ||
| 19. | ALA5251376 | B | Selectivity ratio of IC50 for recombinant human DYRK1B expressed in Sf9 insect cells to IC50 for recombinant human DYRK1A expressed in Sf9 insect cells | Homo sapiens | 48 | cell-based format | Scientific Literature | ||
| 20. | ALA5251377 | B | Selectivity ratio of IC50 for recombinant human GSK-3beta expressed in Sf9 insect cells to IC50 for recombinant human DYRK1A expressed in Sf9 insect cells | Homo sapiens | 48 | cell-based format | Scientific Literature |
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