# | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
---|---|---|---|---|---|---|---|---|---|
1. | ALA1249116 | B | Inhibition of NF-kappaB expressed in HEK293 cells assessed as inhibition of TNF-alpha-induced transcriptional activation at 1 uM treated 24 hrs before TNFalpha challenge by luciferase reporter gene assay relative to control | 18 | cell-based format | Scientific Literature | |||
2. | ALA1249117 | B | Inhibition of AP1 expressed in HEK293 cells assessed as inhibition of PMA-induced transcriptional activation at 1 uM treated 24 hrs before PMA challenge by luciferase reporter gene assay relative to control | 18 | cell-based format | Scientific Literature | |||
3. | ALA1249118 | B | Inhibition of eIF-4E expressed in human FaDu cells assessed as inhibition of translational activation at 1 uM by luciferase reporter gene assay relative to control | 18 | cell-based format | Scientific Literature | |||
4. | ALA4682726 | B | Displacement of [3H]CCPA from human adenosine receptor A1 expressed in CHO cell membranes incubated for 90 mins by radioligand competition assay | Homo sapiens | 35 | cell membrane format | Scientific Literature | ||
5. | ALA4682727 | B | Displacement of [3H]CCPA from adenosine receptor A1 in rat brain cortex membranes incubated for 90 mins by radioligand competition assay | Rattus norvegicus | 28 | cell membrane format | Scientific Literature | ||
6. | ALA4682728 | B | Displacement of [3H]MSX2 from human adenosine receptor A2A expressed in HEK293 cell membranes incubated for 30 mins by radioligand competition assay | Homo sapiens | 35 | cell membrane format | Scientific Literature | ||
7. | ALA4682729 | B | Displacement of [3H]MSX2 from adenosine receptor A2A in rat brain striatum membranes incubated for 30 mins by radioligand competition assay | Rattus norvegicus | 28 | cell membrane format | Scientific Literature | ||
8. | ALA4682730 | B | Displacement of [3H]PSB-603 from human adenosine receptor A2B expressed in CHO cell membranes incubated for 75 mins by radioligand competition assay | Homo sapiens | 31 | cell membrane format | Scientific Literature | ||
9. | ALA4682731 | B | Displacement of [3H]PSB-603 from rat adenosine receptor A2B expressed in CHO cell membranes incubated for 75 mins by radioligand competition assay | Rattus norvegicus | 21 | cell membrane format | Scientific Literature | ||
10. | ALA4682732 | B | Displacement of [3H]PSB-11 from human adenosine receptor A3 expressed in CHO cell membranes incubated for 60 mins by radioligand competition assay | Homo sapiens | 31 | cell membrane format | Scientific Literature | ||
11. | ALA4682733 | B | Displacement of [3H]NECA from rat adenosine receptor A3 expressed in CHO cell membranes incubated for 60 mins by radioligand competition assay | Rattus norvegicus | 16 | cell membrane format | Scientific Literature | ||
12. | ALA4682734 | B | Displacement of [3H]CCPA from adenosine receptor A1 in human brain cortex membranes at 0.1 uM incubated for 90 mins by radioligand competition assay relative to control | Homo sapiens | 7 | cell membrane format | Scientific Literature | ||
13. | ALA4682735 | B | Displacement of [3H]MSX2 from human adenosine receptor A2A expressed in HEK293 cell membranes at 0.1 uM incubated for 30 mins by radioligand competition assay relative to control | Homo sapiens | 10 | cell membrane format | Scientific Literature | ||
14. | ALA4682746 | B | Displacement of [3H]CCPA from adenosine receptor A1 in rat brain cortex membranes at 0.1 uM incubated for 90 mins by radioligand competition assay | Rattus norvegicus | 12 | cell membrane format | Scientific Literature | ||
15. | ALA4682747 | B | Displacement of [3H]MSX2 from adenosine receptor A2A in rat brain striatum membranes at 0.1 uM incubated for 30 mins by radioligand competition assay relative to control | Rattus norvegicus | 15 | cell membrane format | Scientific Literature |