| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA645793 | B | In vitro binding affinity against Alpha-1 adrenergic receptor using [3H]prazosin as radioligand | 20 | protein format | Scientific Literature | |||
| 2. | ALA646863 | B | Affinity for alpha-1 adrenergic receptor in rat was determined by [3H]- prazosin binding assay | 7 | assay format | Scientific Literature | |||
| 3. | ALA645239 | B | Binding affinity against alpha-1 adrenergic receptor | 14 | protein format | Scientific Literature | |||
| 4. | ALA645240 | B | Compound was tested for the binding affinity against alpha-1 adrenergic receptor; NE = 'Not evaluated' | 1 | protein format | Scientific Literature | |||
| 5. | ALA644129 | B | Tested for the Alpha-1 adrenergic receptor affinity in a standard radioligand binding assay with [3H]- prazosin | 7 | protein format | Scientific Literature | |||
| 6. | ALA872367 | B | Binding affinity towards Alpha-1 adrenergic receptor in rat brain using [3H]prazosin | Rattus norvegicus | 9 | tissue-based format | Scientific Literature | ||
| 7. | ALA736789 | F | In vivo effective dose in mice after intraperitoneal administration using standard sound induced seizures assay | Mus musculus | 6 | organism-based format | Scientific Literature | ||
| 8. | ALA877791 | F | ED50 value was calculated by mouse electric shock assay (MES). | Mus musculus | 7 | organism-based format | Scientific Literature | ||
| 9. | ALA747078 | F | Tested for the NMDA antagonist activity using a functional assay, by protection of cultured hippocampus neurons from the toxic effects of extracellularly applied glutamate | 7 | tissue-based format | Scientific Literature | |||
| 10. | ALA752263 | B | Inhibition of [3H]25-6981 binding to N-methyl-D-aspartate glutamate receptor 2B of rat brain | Rattus norvegicus | 13 | assay format | Scientific Literature | ||
| 11. | ALA751683 | B | Binding affinity against NMDA receptor by displacement of [3H]Ro-256981 | 28 | protein complex format | Scientific Literature | |||
| 12. | ALA749674 | B | Binding affinity towards human NR2B receptor | 2 | single protein format | Scientific Literature | |||
| 13. | ALA745941 | F | N-methyl-D-aspartate glutamate receptor antagonistic activity in cell culture(CC)model | 16 | assay format | Scientific Literature | |||
| 14. | ALA745942 | F | Compound was tested for the N-methyl-D-aspartate glutamate receptor antagonistic activity in cell culture(CC)model; NE = 'Not evaluated' | 1 | assay format | Scientific Literature | |||
| 15. | ALA753016 | F | In vitro inhibitory concentration against NMDA responses at cloned NR1A/2A receptors expressed in Xenopus oocytes | Rattus norvegicus | 8 | cell-based format | Scientific Literature | ||
| 16. | ALA752242 | F | In vitro inhibitory concentration against NMDA responses at NR1A/2B receptors expressed in Xenopus oocytes | Rattus norvegicus | 8 | cell-based format | Scientific Literature | ||
| 17. | ALA752250 | F | In vitro inhibitory concentration against NMDA responses at NR1A/2C receptors expressed in Xenopus oocytes | Rattus norvegicus | 8 | cell-based format | Scientific Literature | ||
| 18. | ALA798364 | F | In vitro inhibition of glutamate induced neuronal death in primary cultures of rat hippocampal neurons. | 20 | tissue-based format | Scientific Literature | |||
| 19. | ALA815530 | F | Inhibition of voltage -gated K+ currents was measured by whole cell voltage clamp recordings from dissociated rat superior cervical ganglion neurons at 10 uM | Rattus | 7 | organism-based format | Scientific Literature | ||
| 20. | ALA835748 | B | Selectivity between protection against glutamate-induced neuronal damage and alpha 1 adrenergic affinity | Rattus norvegicus | 14 | assay format | Scientific Literature |
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