| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA751882 | B | Activity against rat cortical and hippocampal membrane strychnine-insensitive N-methyl-D-aspartate glutamate receptor 1 using [3H]-gly | Rattus norvegicus | 11 | tissue-based format | Scientific Literature | ||
| 2. | ALA752489 | B | Ability to compete with [3H]glycine for strychnine-insensitive binding sites on rat cortical and hippocampal membrane | 28 | tissue-based format | Scientific Literature | |||
| 3. | ALA747014 | B | Selectivity ratio for CPP and gly NMDA binding | Rattus norvegicus | 11 | protein complex format | Scientific Literature | ||
| 4. | ALA747511 | B | Activity against rat cortical and hippocampal membrane N-methyl-D-aspartate glutamate receptor 1/2A/2B/2C/2D using [3H]CPP | Rattus norvegicus | 11 | tissue-based format | Scientific Literature | ||
| 5. | ALA749385 | B | Ability to compete with [3H]CCP for rat cortical and hippocampal membrane glutamate binding site. | 17 | tissue-based format | Scientific Literature | |||
| 6. | ALA849492 | B | Ratio of the inhibitory activity against [3H]-CCP for rat cortical and hippocampal membrane glutamate binding site to [3H]glycine for rat cortical and hippocampal membrane binding site. | 16 | tissue-based format | Scientific Literature | |||
| 7. | ALA1952453 | B | Inhibition of human recombinant KAT1 after 20 mins by RP-HPLC analysis | Homo sapiens | 12 | single protein format | Scientific Literature | ||
| 8. | ALA1952454 | B | Ratio of compound IC50 to indole-3-propionic acid IC50 for human recombinant KAT1 | Homo sapiens | 3 | single protein format | Scientific Literature | ||
| 9. | ALA4200085 | F | Agonist activity at human GPR17 expressed in human 1321N1 cells assessed as induction of calcium mobilization after 1 hr by Oregon Green BAPTA-1/AM dye-based fluorescence assay | Homo sapiens | 51 | cell-based format | Scientific Literature | ||
| 10. | ALA4200090 | F | Agonist activity at human GPR17 expressed in human 1321N1 cells assessed as induction of calcium mobilization at >30 uM after 1 hr by Oregon Green BAPTA-1/AM dye-based fluorescence assay relative to control | Homo sapiens | 17 | cell-based format | Scientific Literature | ||
| 11. | ALA4200092 | B | Displacement of [3H]glycine from NMDA receptor in rat cortical and hippocampal membranes | Rattus norvegicus | 7 | assay format | Scientific Literature | ||
| 12. | ALA4200093 | B | Displacement of [3H]CCP from NMDA receptor glutamate binding site in rat cortical and hippocampal membranes | Rattus norvegicus | 5 | assay format | Scientific Literature |
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