| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA631689 | P | Partition coefficient (logP) | 8 | small-molecule physicochemical format | Scientific Literature | |||
| 2. | ALA651677 | B | Binding affinity for rat benzodiazepine receptor inverse agonist site | Rattus norvegicus | 36 | protein complex format | Scientific Literature | ||
| 3. | ALA652368 | B | Concentration to inhibit [3H]flunitrazepam binding to rat cerebral cortical membrane | 15 | assay format | Scientific Literature | |||
| 4. | ALA858255 | B | Binding affinity towards benzodiazepine receptor inverse agonist site by the displacement of [3H]diazepam in rat cerebral cortical membranes. | 51 | cell membrane format | Scientific Literature | |||
| 5. | ALA650289 | B | In vitro inhibition of 3[H]Diazepam binding to Benzodiazepine receptor from rat cerebral cortical membranes | 43 | cell membrane format | Scientific Literature | |||
| 6. | ALA651949 | B | In vitro potency measured against [3H]diazepam at the benzodiazepine receptor in rat | 38 | assay format | Scientific Literature | |||
| 7. | ALA650876 | B | Inhibition of [3H]-diazepam binding to GABA-A benzodiazepine receptor of rat cerebral cortical membranes | Rattus norvegicus | 10 | cell membrane format | Scientific Literature | ||
| 8. | ALA650178 | B | In vitro inhibition of binding to the benzodiazepine receptor in rat cerebral cortical membrane using [3H]diazepam as radioligand | Rattus norvegicus | 18 | cell membrane format | Scientific Literature | ||
| 9. | ALA650075 | B | Inhibition on Benzodiazepine receptor | 43 | protein complex format | Scientific Literature | |||
| 10. | ALA683045 | B | Binding affinity for human recombinant gamma-aminobutyric-acid (GABA) A receptor alpha-6-beta-3-gamma-2 | 144 | protein complex format | Scientific Literature | |||
| 11. | ALA678329 | B | Binding affinity for human recombinant gamma-aminobutyric-acid (GABA) A receptor alpha-1-beta-3-gamma-2 | 146 | protein complex format | Scientific Literature | |||
| 12. | ALA681248 | B | Binding affinity to human recombinant gamma-aminobutyric-acid (GABA) A receptor alpha-2-beta-3-gamma-2 | 136 | protein complex format | Scientific Literature | |||
| 13. | ALA682251 | B | Binding affinity for human recombinant gamma-aminobutyric-acid (GABA) A receptor alpha-3-beta-3-gamma-2 | 146 | protein complex format | Scientific Literature | |||
| 14. | ALA681480 | B | Binding affinity for human recombinant gamma-aminobutyric-acid (GABA) A receptor alpha-5-beta-3-gamma-2 | 149 | protein complex format | Scientific Literature | |||
| 15. | ALA722171 | F | Antagonism of Diazepam (2.5 mg/kg) anticonvulsant effect in mice treated with (pentylenetetrazole) PTZ (80 mg/kg) | Mus musculus | 3 | organism-based format | Scientific Literature | ||
| 16. | ALA722173 | F | Convulsant effect in mice treated with subconvulsant (pentylenetetrazole) PTZ (40 mg/kg) | Mus musculus | 2 | organism-based format | Scientific Literature | ||
| 17. | ALA735984 | F | Antagonism of Diazepam (2.5 mg/kg) anticonvulsant effects in mice treated with PTZ (80 mg/kg) | Mus musculus | 9 | organism-based format | Scientific Literature | ||
| 18. | ALA736885 | F | Convulsant effects in mice treated with PTZ (40 mg/kg) dose | Mus musculus | 10 | organism-based format | Scientific Literature | ||
| 19. | ALA1005398 | B | Displacement of [3H]diazepam from GABAA/BzR in rat brain membrane | Rattus norvegicus | 58 | cell membrane format | Scientific Literature | ||
| 20. | ALA5235567 | B | Binding affinity to human recombinant GABAA alpha1 receptor assessed as inhibition constant incubated for 1 hrs by liquid scintillation counting analysis | Homo sapiens | 21 | single protein format | Scientific Literature |
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