| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA876038 | P | Partition coefficient (logP) | 7 | ALA1122916 | small-molecule physicochemical format | Scientific Literature | ||
| 2. | ALA633363 | P | Solubility in 0.1 M phosphate buffer at pH 7.4 | 7 | ALA1122916 | small-molecule physicochemical format | Scientific Literature | ||
| 3. | ALA633364 | P | Solubility in 0.1 N HCl | 7 | ALA1122916 | small-molecule physicochemical format | Scientific Literature | ||
| 4. | ALA633165 | P | Equilibrium constant (pKa) was determined. | 7 | ALA1122916 | small-molecule physicochemical format | Scientific Literature | ||
| 5. | ALA642474 | B | Log IC50 value was determined against adenosine A1 receptor in rat brain membranes | 16 | ALA1122916 | cell membrane format | Scientific Literature | ||
| 6. | ALA641986 | F | Antagonism of cyclic [3H]AMP accumulation in guinea pig cerebral cortical slices (elicited by 15 uM 2-chloroadenosine at adenosine A2 receptor) | Cavia porcellus | 24 | ALA1123072 | assay format | Scientific Literature | |
| 7. | ALA640601 | B | Inhibitory activity against adenosine A1 receptor in bovine brain membranes | Bos taurus | 1 | ALA1122403 | cell membrane format | Scientific Literature | |
| 8. | ALA640605 | B | Binding affinity against bovine brain adenosine A1 receptor by using N6-[3H]- cyclohexyladenosine | 76 | ALA1122916 | assay format | Scientific Literature | ||
| 9. | ALA640607 | B | Log IC50 value was determined against adenosine A1 receptor in bovine brain membranes | 17 | ALA1122916 | cell membrane format | Scientific Literature | ||
| 10. | ALA640787 | B | Antagonism of binding of 1 nM [3H]cyclohexyladenosine to adenosine A1 receptors on rat cortical membranes | 24 | ALA1123072 | cell membrane format | Scientific Literature | ||
| 11. | ALA639429 | B | Binding affinity against A1 adenosine receptors of the central nervous system | 19 | ALA1123349 | single protein format | Scientific Literature | ||
| 12. | ALA640367 | B | Binding affinity against adenosine A1 receptor using [3H]-CHA or [3H]PIA as radioligand | 44 | ALA1125572 | single protein format | Scientific Literature | ||
| 13. | ALA636644 | B | Inhibition of [3H]CHA binding to Adenosine A1 receptor in rat brain membranes | Rattus norvegicus | 5 | ALA1124797 | cell membrane format | Scientific Literature | |
| 14. | ALA644772 | B | Binding affinity against A2 adenosine receptors of the central nervous system | 19 | ALA1123349 | protein format | Scientific Literature | ||
| 15. | ALA645326 | B | Binding affinity against adenosine A2 receptor using [3H]- NECA as radioligand | 44 | ALA1125572 | protein format | Scientific Literature | ||
| 16. | ALA645332 | B | Ratio of A2 to A1. | 49 | ALA1125572 | protein format | Scientific Literature | ||
| 17. | ALA638324 | B | Selectivity ratio was expressed as the ratio of binding affinity towards Adenosine A2 receptor to that of Adenosine A1 receptor in rat | 19 | ALA1123349 | assay format | Scientific Literature | ||
| 18. | ALA664964 | F | log(1000/IC50 determined from bovine brain membrane) expressed as potency | Bos taurus | 1 | ALA1122916 | organism-based format | Scientific Literature | |
| 19. | ALA666570 | F | log(1000/IC50 determined from bovine brain membrane) expressed as potency | Bos taurus | 1 | ALA1122916 | organism-based format | Scientific Literature | |
| 20. | ALA782817 | F | Inhibitory activity against rat brain membranes. | Rattus norvegicus | 1 | ALA1122916 | organism-based format | Scientific Literature |
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