| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA1613855 | F | PUBCHEM_BIOASSAY: Late stage results from the probe development effort to identify inhibitors of the protein methylesterase PME-1: Gel-based Activity-Based Protein Profiling (ABPP) IC50: Purified enzyme. (Class of assay: confirmatory) [Related pubchem assays: 2143 (Summary AID (PME-1 inhibitors)), 2130 (PME-1 inhibitors in singlate), 2174 (LYPLA1 inhibitors in singlate), 2177 (LYPLA2 inhibitors in singlate), 2171 (PME-1 inhibitors in triplicate), 2291 (PME-1 inhibitors in singlate), 2233 (LYPLA1 inhibitors in triplicate), 2232 (LYPLA2 inhibitors in triplicate)] | Homo sapiens | 6 | assay format | PubChem BioAssays | ||
| 2. | ALA1738413 | U | PUBCHEM_BIOASSAY: Late stage results from the probe development effort to identify inhibitors of the protein methylesterase PME-1: Gel-based Activity-Based Protein Profiling (ABPP) IC50. (Class of assay: confirmatory) [Related pubchem assays (depositor defined):AID2130, AID2143, AID2171, AID2174, AID2177, AID2232, AID2233, AID2291, AID463090, AID463091, AID463124, AID463130, AID463131, AID463132, AID463146, AID463149] Panel member name: PME-1 Assay Panel member description: Inhibition of endogenously expressed PME-1 | 26 | assay format | PubChem BioAssays | |||
| 3. | ALA2212398 | B | Inhibition of prolyl endopeptidase binding to FP-rhodamine in mouse brain soluble proteome at 50 uM after 30 mins by fluorescence polarization activity-based protein profiling assay relative to control | Mus musculus | 2 | tissue-based format | Scientific Literature | ||
| 4. | ALA2212400 | B | Inhibition of PME1 binding to FP-rhodamine in mouse brain soluble proteome at 20 uM after 30 mins by fluorescence polarization activity-based protein profiling assay relative to control | Mus musculus | 8 | tissue-based format | Scientific Literature |
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