| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA751877 | B | Relative affinity evaluated for Opioid receptor mu 1 | Cavia porcellus | 6 | ALA1135939 | single protein format | Scientific Literature | |
| 2. | ALA752039 | B | Binding affinity using guinea pig brain membrane preparations, towards Opioid receptor mu 1 using [3H]- DAMGO as radioligand | Cavia porcellus | 6 | ALA1135939 | assay format | Scientific Literature | |
| 3. | ALA758250 | B | Relative affinity evaluated for Opioid receptor kappa 1 | Cavia porcellus | 6 | ALA1135939 | single protein format | Scientific Literature | |
| 4. | ALA758257 | B | Binding affinity using guinea pig brain membrane preparations, towards Opioid receptor kappa 1 using [3H]- U-69,593 as radioligand | Cavia porcellus | 6 | ALA1135939 | assay format | Scientific Literature | |
| 5. | ALA756037 | B | Relative affinity evaluated for Opioid receptor delta 1 | Cavia porcellus | 6 | ALA1135939 | single protein format | Scientific Literature | |
| 6. | ALA857861 | B | Binding affinity using guinea pig brain membrane preparations, towards Opioid receptor delta 1 using [3H]DPDPE as radioligand | Cavia porcellus | 6 | ALA1135939 | assay format | Scientific Literature | |
| 7. | ALA818456 | F | % maximum inhibition is elicited when the response reaches plateau, calculated regarding electrically induced contraction in guinea pig ileum as 100% (P < 0.001) | Cavia porcellus | 3 | ALA1135939 | organism-based format | Scientific Literature | |
| 8. | ALA843391 | F | Relative inhibitory activity expressed as the percentage of the maximum inhibition by the compound against that of morphine | Cavia porcellus | 12 | ALA1135939 | organism-based format | Scientific Literature | |
| 9. | ALA841375 | F | Relative potency expressed as the percentage of the pD2 value against that of morphine | Cavia porcellus | 11 | ALA1135939 | organism-based format | Scientific Literature | |
| 10. | ALA841899 | F | activity evaluated by its ability to inhibit the electrically induced twitch contraction in guinea pig ileum, which is reversed by naloxone (300 nM) | Cavia porcellus | 3 | ALA1135939 | organism-based format | Scientific Literature | |
| 11. | ALA2399173 | B | Agonist activity at opioid receptor in guinea pig ileum assessed as inhibition of electrically-induced twitch at 100 pM to 30 uM relative to morphine | Cavia porcellus | 7 | ALA2396537 | tissue-based format | Scientific Literature | |
| 12. | ALA4380064 | B | Displacement of [3H]prazosin from human recombinant adrenergic alpha-1A receptor expressed in CHO cell membranes at 100 nM incubated for 60 mins relative to control | Homo sapiens | 5 | ALA4376854 | cell-based format | Scientific Literature | |
| 13. | ALA4380065 | B | Displacement of [3H]prazosin from human recombinant adrenergic alpha-1B receptor expressed in CHO cell membranes at 100 nM incubated for 60 mins relative to control | Homo sapiens | 5 | ALA4376854 | cell-based format | Scientific Literature | |
| 14. | ALA4380066 | B | Displacement of [3H]prazosin from human recombinant adrenergic alpha-1D receptor expressed in CHO cell membranes at 100 nM incubated for 60 mins relative to control | Homo sapiens | 5 | ALA4376854 | cell-based format | Scientific Literature | |
| 15. | ALA4380067 | B | Displacement of [3H]RX 821002 from human recombinant adrenergic alpha-2A receptor expressed in CHO cell membranes at 100 nM incubated for 60 mins relative to control | Homo sapiens | 5 | ALA4376854 | cell-based format | Scientific Literature | |
| 16. | ALA4380068 | B | Displacement of [3H]RX 821002 from human recombinant adrenergic alpha-2B receptor expressed in CHO cell membranes at 100 nM incubated for 60 mins relative to control | Homo sapiens | 5 | ALA4376854 | cell-based format | Scientific Literature | |
| 17. | ALA4380069 | B | Displacement of [3H]DADLE from human recombinant delta opioid receptor expressed in rat Chem-1 (RBL) cell membranes at 100 nM incubated for 60 mins relative to control | Homo sapiens | 5 | ALA4376854 | cell-based format | Scientific Literature | |
| 18. | ALA4380070 | B | Displacement of [3H]U69,593 from human recombinant kappa opioid receptor expressed in rat RBL cell membranes at 100 nM incubated for 60 mins relative to control | Homo sapiens | 5 | ALA4376854 | cell-based format | Scientific Literature | |
| 19. | ALA4380071 | B | Displacement of [3H]DAMGO from human recombinant mu opioid receptor expressed in HEK293 cell membranes at 100 nM incubated for 60 mins relative to control | Homo sapiens | 5 | ALA4376854 | cell-based format | Scientific Literature | |
| 20. | ALA4380072 | B | Displacement of radioligand from ORL1 (unknown origin) at 100 nM incubated for 120 mins relative to control | Homo sapiens | 5 | ALA4376854 | single protein format | Scientific Literature |
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