| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA675743 | B | Binding affinity at dopamine receptor D2 on Sf9 cells by [125I]IABN displacement. | 21 | ALA1146691 | cell-based format | Scientific Literature | ||
| 2. | ALA674591 | B | Binding affinity at dopamine receptor D3 on Sf9 cells by [125I]IABN displacement. | 21 | ALA1146691 | cell-based format | Scientific Literature | ||
| 3. | ALA810659 | B | Inhibition of [3H](+)-pentazocine binding to Sigma opioid receptor of guiena pig brain membrane | Cavia porcellus | 14 | ALA1146691 | assay format | Scientific Literature | |
| 4. | ALA808105 | B | Inhibition of [3H](+)-DTG binding to Sigma opioid receptor (type 2) of rat liver membranes in the presence of (+)-pentazocine | Rattus norvegicus | 14 | ALA1146691 | cell membrane format | Scientific Literature | |
| 5. | ALA845651 | B | Ratio of Ki of sigma-1 receptor versus Ki of sigma-2 receptor | 5 | ALA1146691 | single protein format | Scientific Literature | ||
| 6. | ALA931110 | B | Binding affinity to sigma 2 receptor in rat liver membrane by saturation analysis | Rattus norvegicus | 3 | ALA1143158 | cell membrane format | Scientific Literature | |
| 7. | ALA931108 | B | Selectivity for rat sigma 2 receptor over rat sigma1 receptor | Rattus norvegicus | 2 | ALA1143158 | assay format | Scientific Literature | |
| 8. | ALA3238651 | B | Selectivity ratio of Ki for sigma-1 opioid receptor (unknown origin) to Ki for sigma-2 opioid receptor (unknown origin) | Homo sapiens | 16 | ALA3232965 | assay format | Scientific Literature | |
| 9. | ALA3238652 | B | Binding affinity to sigma-1 opioid receptor (unknown origin) | Homo sapiens | 20 | ALA3232965 | single protein format | Scientific Literature | |
| 10. | ALA3238653 | B | Binding affinity to sigma-2 opioid receptor (unknown origin) | Homo sapiens | 20 | ALA3232965 | assay format | Scientific Literature | |
| 11. | ALA3271176 | P | Lipophilicity, log P of the compound | 7 | ALA3259688 | small-molecule physicochemical format | Scientific Literature | ||
| 12. | ALA3271543 | B | Displacement of 5-bromo-N-(4-(3,4-dihydro-6,7-dimethoxyisoquinolin-2(1H)-yl)butyl)-2,3-dimethoxybenzamide from sigma-1 receptor in mouse EMT6 cell membranes after 60 mins by Scatchard plot analysis | Mus musculus | 3 | ALA3259688 | cell-based format | Scientific Literature | |
| 13. | ALA3271544 | B | Displacement of 5-bromo-N-(4-(3,4-dihydro-6,7-dimethoxyisoquinolin-2(1H)-yl)butyl)-2,3-dimethoxybenzamide from sigma-2 receptor in mouse EMT6 cell membranes after 60 mins by Scatchard plot analysis | Mus musculus | 3 | ALA3259688 | cell-based format | Scientific Literature | |
| 14. | ALA3271545 | B | Selectivity ratio of Ki for sigma-1 receptor in mouse EMT6 cell membranes to Ki for sigma-2 receptor in mouse EMT6 cell membranes | Mus musculus | 3 | ALA3259688 | cell-based format | Scientific Literature | |
| 15. | ALA4148655 | B | Binding affinity to sigma-1 receptor (unknown origin) | Homo sapiens | 8 | ALA4145543 | single protein format | Scientific Literature | |
| 16. | ALA4148656 | B | Binding affinity to sigma-2 receptor (unknown origin) | Homo sapiens | 8 | ALA4145543 | single protein format | Scientific Literature | |
| 17. | ALA4733425 | B | Antagonist activity at sigma 2 receptor in human MCF7 cells assessed as reduction in intracellular calcium release at 30 uM incubated for 3 hrs by Fluo-3 AM dye based confocal laser scanning microscopy | Homo sapiens | 5 | ALA4732061 | cell-based format | Scientific Literature |
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