# | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
---|---|---|---|---|---|---|---|---|---|
1. | ALA652562 | B | In vitro inhibition of [3H]diazepam binding to benzodiazepine receptor in rat cerebral cortical membrane | 48 | ALA1122149 | cell membrane format | Scientific Literature | ||
2. | ALA3051423 | A | Inhibition of Oryctolagus cuniculus (rabbit) AOX in liver cytosol at IC50 concentration | Oryctolagus cuniculus | 17 | ALA3045711 | tissue-based format | Scientific Literature | |
3. | ALA3051424 | B | Inhibition of xanthine oxidase at IC50 concentration | 20 | ALA3045711 | assay format | Scientific Literature | ||
4. | ALA3051429 | B | Inhibition of xanthine oxidase | 30 | ALA3045711 | assay format | Scientific Literature | ||
5. | ALA3051430 | A | Inhibition of Oryctolagus cuniculus (rabbit) AOX in liver cytosol | Oryctolagus cuniculus | 30 | ALA3045711 | tissue-based format | Scientific Literature | |
6. | ALA3051431 | B | Inhibition of Agaricus bisporus (mushroom) tyrosinase | Agaricus bisporus | 30 | ALA3045711 | single protein format | Scientific Literature | |
7. | ALA3051195 | F | Nematicidal activity against Meloidogyne incognita (root-knot nematode) juveniles J2 assessed as paralysis after 1 day | Meloidogyne incognita | 17 | ALA3045343 | organism-based format | Scientific Literature | |
8. | ALA3051196 | F | Nematicidal activity against Meloidogyne incognita (root-knot nematode) juveniles J2 assessed as paralysis after 1 hr | Meloidogyne incognita | 17 | ALA3045343 | organism-based format | Scientific Literature | |
9. | ALA3240837 | B | Inhibition of NorA in fluoroquinolone-resistant Staphylococcus aureus 1199B assessed as potentiation of 4 ug/ml of ciprofloxacin MIC at 100 ug/ml after 24 hrs by microdilution method | Staphylococcus aureus | 135 | ALA3232989 | assay format | Scientific Literature | |
10. | ALA3240840 | A | Toxicity in Staphylococcus aureus ATCC 25923 after 24 hrs by microdilution method | Staphylococcus aureus | 129 | ALA3232989 | organism-based format | Scientific Literature | |
11. | ALA3240841 | A | Toxicity in fluoroquinolone-resistant Staphylococcus aureus 1199B expressing NorA after 24 hrs by microdilution method | Staphylococcus aureus | 44 | ALA3232989 | organism-based format | Scientific Literature | |
12. | ALA3637356 | B | Inhibition of Mycobacterium tuberculosis MTCC 300 DAH7PS expressed in Escherichia coli BL21 (DE3) using 25 to 125 uM PEP/100 uM E4P as substrate up to 50 nM by spectrophotometric analysis | Mycobacterium tuberculosis | 5 | ALA3632512 | assay format | Scientific Literature | |
13. | ALA3637357 | B | Inhibition of Mycobacterium tuberculosis MTCC 300 DAH7PS expressed in Escherichia coli BL21 (DE3) using 25 to 125 uM PEP/100 uM E4P as substrate at 10 uM by spectrophotometric analysis relative to control | Mycobacterium tuberculosis | 6 | ALA3632512 | assay format | Scientific Literature | |
14. | ALA3637358 | B | Inhibition of Mycobacterium tuberculosis MTCC 300 DAH7PS expressed in Escherichia coli BL21 (DE3) using 25 to 125 uM PEP/100 uM E4P as substrate by spectrophotometric analysis | Mycobacterium tuberculosis | 6 | ALA3632512 | assay format | Scientific Literature | |
15. | ALA4342201 | B | Inhibition of NO711 binding to mouse GAT1 expressed in HEK293 cell membranes assessed as residual binding at 1 uM incubated for 4 hrs in presence of NO711 by LC-ESI-MS/MS analysis relative to control | Mus musculus | 247 | ALA4340561 | cell-based format | Scientific Literature | |
16. | ALA4401740 | B | Inhibition of mouse GAT-1 assessed as percentage of remaining specific binding of NO711 at 1 uM after 4 hrs by LC-ESI-MS/ms analysis relative to control | Mus musculus | 176 | ALA4400545 | single protein format | Scientific Literature | |
17. | ALA4422579 | B | Inhibition of StrepTag-tagged human SARM1 TIR (561 to 724 residues) expressed in HEK293T cells assessed as reduction in NADase activity in presence of NAD+ incubated for 60 mins by HPLC analysis | Homo sapiens | 26 | ALA4421736 | cell-based format | Patent Bioactivity Data | |
18. | ALA4422585 | B | Substrate activity at StrepTag-tagged human SARM1 TIR (561 to 724 residues) expressed in HEK293T cells assessed as increase in in NADase activity in presence of NAD+ incubated for 60 mins by HPLC analysis | Homo sapiens | 9 | ALA4421736 | cell-based format | Patent Bioactivity Data |