# | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
---|---|---|---|---|---|---|---|---|---|
1. | ALA751111 | F | Antagonist activity against recombinant rat receptor P2X purinoceptor 2 (P2X2) at 10 uM, expressed in Xenopus oocytes | 7 | ALA1135773 | cell-based format | Scientific Literature | ||
2. | ALA751112 | F | The compound was evaluated for antagonist activity against recombinant rat receptor P2X purinoceptor 2 (P2X2) at 30 uM, expressed in Xenopus oocytes | 2 | ALA1135773 | cell-based format | Scientific Literature | ||
3. | ALA751802 | F | The compound was evaluated for antagonist activity against recombinant rat receptor P2X purinoceptor 2 (P2X4) at 30 uM, expressed in Xenopus oocytes | 2 | ALA1135773 | cell-based format | Scientific Literature | ||
4. | ALA857685 | F | The compound was evaluated for antagonist activity against recombinant rat P2X purinoceptor 2 (P2X2) at 10 uM | 1 | ALA1135773 | assay format | Scientific Literature | ||
5. | ALA754946 | F | Inhibition of inward ion current elicited by ATP at P2X2 receptor expressed in Xenopus oocytes; IA means inactive | Rattus norvegicus | 2 | ALA1134335 | cell-based format | Scientific Literature | |
6. | ALA754947 | F | Inhibition of inward ion current elicited by ATP at P2X2 receptor expressed in Xenopus oocytes | Rattus norvegicus | 10 | ALA1134335 | cell-based format | Scientific Literature | |
7. | ALA759525 | F | The compound was evaluated for antagonist activity against recombinant rat P2X purinoceptor 2 (P2X2) at 30 uM | 1 | ALA1135773 | assay format | Scientific Literature | ||
8. | ALA760168 | F | The compound was evaluated for antagonist activity against recombinant rat receptor P2X purinoceptor 2 (P2X2) at 10 uM, expressed in Xenopus oocytes | 1 | ALA1135773 | cell-based format | Scientific Literature | ||
9. | ALA872172 | F | Inhibitory concentration against rat P2X purinoceptor 2 expressed in Xenopus laevis oocytes | Rattus norvegicus | 1 | ALA1140384 | cell-based format | Scientific Literature | |
10. | ALA901771 | B | Activity at rat P2X2 receptor at 10 uM | Rattus norvegicus | 2 | ALA1138274 | single protein format | Scientific Literature | |
11. | ALA1680807 | F | Antagonist activity against rat P2X2 receptor expressed in Xenopus laevis oocyte assessed as inhibition of alpha, beta-meATP-induced inward current by two-electrode voltage-clamp electrophysiology | Rattus norvegicus | 61 | ALA1671813 | assay format | Scientific Literature | |
12. | ALA1680808 | F | Antagonist activity against rat P2X2 receptor expressed in Xenopus laevis oocyte assessed as inhibition of alpha, beta-meATP-induced inward current at 100 nM by two-electrode voltage-clamp electrophysiology | Rattus norvegicus | 4 | ALA1671813 | assay format | Scientific Literature | |
13. | ALA1680827 | F | Antagonist activity against rat P2X2 receptor expressed in Xenopus laevis oocyte assessed as maximum current amplitude by two-electrode voltage-clamp electrophysiology | Rattus norvegicus | 1 | ALA1671813 | assay format | Scientific Literature | |
14. | ALA1680828 | F | Antagonist activity against rat P2X2 receptor expressed in Xenopus laevis oocyte assessed as maximum alpha, beta-meATP-induced inward current by two-electrode voltage-clamp electrophysiology in presence of 10 uM ATP | Rattus norvegicus | 1 | ALA1671813 | assay format | Scientific Literature | |
15. | ALA2400255 | B | Activity at rat recombinant purinergic P2X2 receptor expressed in Xenopus oocytes assessed as effect on ATP-induced activation at 3 uM by two-electrode voltage clamp technique relative to control | Rattus norvegicus | 1 | ALA2396604 | cell-based format | Scientific Literature | |
16. | ALA2427309 | B | Inhibition of rat purinergic receptor P2X subunit-2 expressed in Xenopus laevis oocytes assessed as inhibition of ATP-induced current at 3 uM by two-electrode voltage clamp method | Rattus norvegicus | 2 | ALA2424574 | cell-based format | Scientific Literature | |
17. | ALA4031268 | B | Inhibition of rat P2X2 receptor expressed in xenopus lavies oocytes assessed as inhibition of ATP-induced peak current at 3 mM by two electrode voltage clamp | Rattus norvegicus | 1 | ALA4028862 | cell-based format | Scientific Literature | |
18. | ALA4153222 | B | Antagonist activity at wild type His6 tagged rat P2X1 receptor expressed in Xenopus laevis oocytes assessed as inhibition of alphabeta-me ATP-induced calcium flux at -60 mV holding potential by two electrode voltage clamp method | Rattus norvegicus | 1 | ALA4152208 | cell-based format | Scientific Literature | |
19. | ALA4714127 | B | Antagonist activity at rat P2X2 receptor expressed in Xenopus laevis oocytes assessed as reduction in ATP-induced channel currents at 100 uM by TEVC electrophysiology assay relative to control | Rattus norvegicus | 1 | ALA4706687 | cell-based format | Scientific Literature |