| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA856245 | F | Inhibitory concentration against human gastric inhibitory polypeptide receptor (hGIP) mediated cAMP accumulation | Homo sapiens | 1 | tissue-based format | Scientific Literature | ||
| 2. | ALA911155 | B | Inhibition of GIP receptor at 10 uM | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 3. | ALA1924544 | F | Inhibition of human GIP receptor by cAMP assay | Homo sapiens | 6 | single protein format | Scientific Literature | ||
| 4. | ALA1925822 | F | Antagonist activity at human GIP receptor assessed as inhibition of cAMP production | Homo sapiens | 1 | assay format | Scientific Literature | ||
| 5. | ALA1937454 | B | Displacement of [125I]GIP from human GIPR | Homo sapiens | 4 | single protein format | Scientific Literature | ||
| 6. | ALA890127 | F | Antagonist activity at human GIP receptor transfected in CHO cells assessed as inhibition of glucagon-induced cAMP accumulation | Homo sapiens | 16 | cell-based format | Scientific Literature | ||
| 7. | ALA2161796 | F | Agonist activity at human GIP receptor expressed in HEK293 cells assessed as stimulation of cAMP levels incubated for 6 hrs by multiple response element/cAMP response element (MRE/CRE)-driven reporter gene assay | Homo sapiens | 2 | cell-based format | Scientific Literature | ||
| 8. | ALA940051 | F | Agonist activity at human GIP receptor expressed in BHK cells assessed as cAMP accumulation | Homo sapiens | 1 | cell-based format | Scientific Literature | ||
| 9. | ALA945218 | B | Binding affinity against human GIP | Homo sapiens | 14 | single protein format | Scientific Literature | ||
| 10. | ALA995931 | B | Binding affinity to human recombinant GIPR expressed in BHK cells by membrane filter assay | Homo sapiens | 12 | cell-based format | Scientific Literature | ||
| 11. | ALA973452 | B | Displacement of [125I]porcine GIP from human recombinant GIPR receptor expressed in BHK cells by scintillation proximity assay | Homo sapiens | 30 | cell-based format | Scientific Literature | ||
| 12. | ALA977342 | B | Binding affinity to human cloned GIPR expressed in BHK cells | Homo sapiens | 27 | cell-based format | Scientific Literature | ||
| 13. | ALA1050755 | F | Agonist activity at GIPR | 1 | assay format | Scientific Literature | |||
| 14. | ALA1648236 | F | Antagonist activity at human GIPR expressed in CHO cells assessed as inhibition of glucagon-induced cAMP accumulation | Homo sapiens | 19 | cell-based format | Scientific Literature | ||
| 15. | ALA1648901 | F | Antagonist activity at human GIPR expressed in CHO cells assessed as inhibition of glucagon-induced cAMP accumulation at 10 uM | Homo sapiens | 22 | cell-based format | Scientific Literature | ||
| 16. | ALA2160603 | F | Antagonist activity at human GIPR expressed in CHO cells assessed as inhibition of glucagon-induced cAMP accumulation preincubated for 30 mins prior to glucagon challenge measured after 30 mins post glucagon challenge by liquid scintillation counter | Homo sapiens | 21 | cell-based format | Scientific Literature | ||
| 17. | ALA3242379 | F | Antagonist activity at human GIPR assessed as inhibition of cAMP production | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 18. | ALA3362655 | F | Antagonist activity at human GIP receptor expressed in HEK293 cells by IP4 HTRF EFC cAMP/summary (Abse5) assay | Homo sapiens | 1 | cell-based format | Scientific Literature | ||
| 19. | ALA3620261 | F | Antagonist activity against human glucose dependent insulinotropic peptide receptor by cAMP accumulation assay | Homo sapiens | 5 | single protein format | Scientific Literature | ||
| 20. | ALA4124802 | F | Agonist activity at human GIP receptor expressed in HEK293 cells assessed as cAMP accumulation after 30 mins by HTRF assay | Homo sapiens | 16 | cell-based format | Scientific Literature |
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