# | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
---|---|---|---|---|---|---|---|---|---|
1. | ALA861844 | F | Agonist potency at human GPR40 expressed in CHO cells | Homo sapiens | 38 | cell-based format | Scientific Literature | ||
2. | ALA861845 | F | Agonist potency at human GPR40 expressed in CHO cells relative to standard by luciferase reporter gene assay | Homo sapiens | 38 | cell-based format | Scientific Literature | ||
3. | ALA943950 | F | Activity at FFAR1 expressed in HEK-EM293 cells assessed as calcium influx relative to GW-9508 by FLIPR assay | 12 | cell-based format | Scientific Literature | |||
4. | ALA943951 | F | Agonist activity at FFAR1 expressed in HEK-EM293 cells assessed as calcium influx by FLIPR assay | 20 | cell-based format | Scientific Literature | |||
5. | ALA943952 | F | Antagonist activity at FFAR1 expressed in HEK-EM293 cells assessed as inhibition calcium influx by FLIPR assay | 2 | cell-based format | Scientific Literature | |||
6. | ALA943953 | F | Antagonist activity at FFAR1 expressed in HEK-EM293 cells assessed as linoleic acid-stimulated calcium influx after 30 mins by FLIPR assay | 1 | cell-based format | Scientific Literature | |||
7. | ALA944876 | F | Activity at FFAR1 R183A mutant expressed in HEK-EM293 cells assessed as calcium influx by FLIPR assay | Homo sapiens | 2 | cell-based format | Scientific Literature | ||
8. | ALA944877 | F | Activity at FFAR1 H86F mutant expressed in HEK-EM293 cells assessed as calcium influx by FLIPR assay | Homo sapiens | 2 | cell-based format | Scientific Literature | ||
9. | ALA944878 | F | Activity at FFAR1 H137F mutant expressed in HEK-EM293 cells assessed as calcium influx by FLIPR assay | Homo sapiens | 2 | cell-based format | Scientific Literature | ||
10. | ALA944879 | F | Activity at FFAR1 L186F mutant expressed in HEK-EM293 cells assessed as calcium influx by FLIPR assay | Homo sapiens | 2 | cell-based format | Scientific Literature | ||
11. | ALA944880 | F | Activity at FFAR1 N244A mutant expressed in HEK-EM293 cells assessed as calcium influx by FLIPR assay | Homo sapiens | 2 | cell-based format | Scientific Literature | ||
12. | ALA944881 | F | Activity at FFAR1 expressed in HEK-EM293 cells assessed as calcium influx by FLIPR assay | 2 | cell-based format | Scientific Literature | |||
13. | ALA2027152 | F | Agonist activity at human GR40 receptor expressed in CHO cells assessed as increase in intracellular calcium concentration after 90 secs by FLIPR assay in presence of 0.1% BSA | Homo sapiens | 26 | cell-based format | Scientific Literature | ||
14. | ALA2027153 | B | Displacement of 3-[4-({2',6'-dimethyl-6-[(4-[3H])-phenylmethoxy]biphenyl-3-yl}methoxy)phenyl] propanoic acid from human GPR40 receptor expressed in CHO cells after 90 mins by scintillation counting in presence of 0.2% BSA | Homo sapiens | 26 | cell-based format | Scientific Literature | ||
15. | ALA2027155 | F | Agonist activity at human GR40 receptor expressed in CHO cells assessed as increase in intracellular calcium concentration at 10 uM after 90 secs by FLIPR assay in presence of 0.1% BSA relative to control | Homo sapiens | 2 | cell-based format | Scientific Literature | ||
16. | ALA2027156 | F | Agonist activity at human GR40 receptor expressed in CHO cells assessed as increase in intracellular calcium concentration at 1 uM after 90 secs by FLIPR assay in presence of 0.1% BSA relative to control | Homo sapiens | 2 | cell-based format | Scientific Literature | ||
17. | ALA890929 | F | Agonist activity at GPR40 receptor | Homo sapiens | 34 | assay format | Scientific Literature | ||
18. | ALA890932 | F | Agonist activity at GPR40 receptor expressed in CHO cells by reporter gene assay | Homo sapiens | 34 | cell-based format | Scientific Literature | ||
19. | ALA905041 | F | Agonist activity at human GPR40 expressed in HEK293 cells assessed as effect on calcium flux | Homo sapiens | 21 | cell-based format | Scientific Literature | ||
20. | ALA905042 | F | Agonist activity at human GPR40 expressed in HEK293 cells assessed as calcium flux response relative to linoleic acid | Homo sapiens | 21 | cell-based format | Scientific Literature |