# | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
---|---|---|---|---|---|---|---|---|---|
1. | ALA1166722 | B | Binding affinity to GAT2 | 2 | ALA1165889 | single protein format | Scientific Literature | ||
2. | ALA1647451 | B | Inhibition of GAT2 | 1 | ALA1641586 | single protein format | Scientific Literature | ||
3. | ALA1663479 | B | Inhibition of [3H]GABA uptake at GAT2 expressed in HEK cells | 17 | ALA1649378 | cell-based format | Scientific Literature | ||
4. | ALA1663480 | B | Inhibition of [3H]GABA uptake at GAT2 expressed in HEK cells at 100 uM | 6 | ALA1649378 | cell-based format | Scientific Literature | ||
5. | ALA2208546 | B | Inhibition of human GAT2 expressed in tcA201 cells assessed as inhibition of [3H]GABA uptake at 1 mM after 3 mins by scintillation counting | Homo sapiens | 1 | ALA2203122 | cell-based format | Scientific Literature | |
6. | ALA2417029 | B | Inhibition of human GAT2 transfected in CHO cells assessed as [3H]GABA uptake after 20 mins by liquid scintillation counting analysis | Homo sapiens | 3 | ALA2413054 | cell-based format | Scientific Literature | |
7. | ALA2417033 | B | Inhibition of human GAT2 transfected in CHO cells assessed as [3H]GABA uptake at 100 uM after 20 mins by liquid scintillation counting analysis | Homo sapiens | 8 | ALA2413054 | cell-based format | Scientific Literature | |
8. | ALA3363497 | B | Inhibition of human GAT2 transfected in CHO cells assessed as [3H]GABA uptake after 20 mins by liquid scintillation counting analysis | Homo sapiens | 5 | ALA3351485 | cell-based format | Scientific Literature | |
9. | ALA3363503 | B | Inhibition of human GAT2 transfected in CHO cells assessed as [3H]GABA uptake at 100 uM after 20 mins by liquid scintillation counting analysis | Homo sapiens | 2 | ALA3351485 | cell-based format | Scientific Literature | |
10. | ALA4031698 | B | Inhibition of human GAT2 expresses in tsA201 cells assessed as reduction in [3H]GABA uptake after 3 mins by scintillation counting method | Homo sapiens | 32 | ALA4028872 | cell-based format | Scientific Literature | |
11. | ALA4267185 | B | Inhibition of human GAT2 expressed in CHO cells assessed as reduction in [3H]GABA uptake at 100 uM after 20 mins by liquid scintillation counting analysis relative to control | Homo sapiens | 8 | ALA4265902 | cell-based format | Scientific Literature | |
12. | ALA4398053 | B | Inhibition of human GAT2 expressed in Flp-In CHO cells assessed as reduction in [3H]GABA uptake incubated for 3 mins by liquid scintillation counting method | Homo sapiens | 11 | ALA4396887 | cell-based format | Scientific Literature | |
13. | ALA4398057 | B | Inhibition of human GAT2 expressed in Flp-In CHO cells assessed as reduction in [3H]GABA uptake at 100 uM incubated for 3 mins by liquid scintillation counting method relative to control | Homo sapiens | 10 | ALA4396887 | cell-based format | Scientific Literature | |
14. | ALA4767580 | B | Inhibition of human GTA2 receptor expressed in tsA201 cells assessed as inhibition of [3H]GABA uptake by liquid scintillation method | Homo sapiens | 1 | ALA4765247 | cell-based format | Scientific Literature | |
15. | ALA5098965 | B | Antagonist activity at human GAT2 expressed in CHO cells assessed as [3H]GABA uptake at 50 uM incubated for 3 mins by top-counter microplate scintillation counter assay | Homo sapiens | 1 | ALA5096209 | cell-based format | Scientific Literature |