# | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
---|---|---|---|---|---|---|---|---|---|
1. | ALA869921 | B | Inhibition of lysophospholipase D autotaxin | Homo sapiens | 14 | ALA1148595 | single protein format | Scientific Literature | |
2. | ALA865903 | B | Inhibition of recombinant ATX from transfected HEK293 cells | Homo sapiens | 12 | ALA1149458 | cell-based format | Scientific Literature | |
3. | ALA887356 | B | Inhibition of human recombinant ATX at 1 uM after 16 hrs | Homo sapiens | 39 | ALA1144604 | single protein format | Scientific Literature | |
4. | ALA887357 | B | Inhibition of human recombinant ATX at 10 uM after 16 hrs | Homo sapiens | 39 | ALA1144604 | single protein format | Scientific Literature | |
5. | ALA887358 | B | Inhibition of human recombinant ATX at 100 uM after 16 hrs | Homo sapiens | 39 | ALA1144604 | single protein format | Scientific Literature | |
6. | ALA933171 | B | Inhibition of autotaxin assessed as residual enzyme activity at 1 uM relative to control | 20 | ALA1142314 | single protein format | Scientific Literature | ||
7. | ALA933172 | B | Inhibition of autotaxin assessed as residual enzyme activity at 10 uM relative to control | 20 | ALA1142314 | single protein format | Scientific Literature | ||
8. | ALA933173 | B | Inhibition of autotaxin assessed as residual enzyme activity at 100 uM relative to control | 20 | ALA1142314 | single protein format | Scientific Literature | ||
9. | ALA921041 | B | Inhibition of human autotaxin expressed in MDA-MB-435 cells assessed as fluorescent lysophosphatidyl choline analog hydrolysis at 10 uM | Homo sapiens | 146 | ALA1143995 | cell-based format | Scientific Literature | |
10. | ALA978912 | B | Activity of human autotaxin in human MBA-MBA-435 cells assessed as effect on enzyme-mediated of FS3 hydrolysis at 0.1 uM | Homo sapiens | 35 | ALA1138619 | cell-based format | Scientific Literature | |
11. | ALA978913 | B | Activity of human autotaxin in human MBA-MBA-435 cells assessed as effect on enzyme-mediated of FS3 hydrolysis at 1 uM | Homo sapiens | 35 | ALA1138619 | cell-based format | Scientific Literature | |
12. | ALA978914 | B | Activity of human autotaxin in human MBA-MBA-435 cells assessed as effect on enzyme-mediated of FS3 hydrolysis at 10 uM | Homo sapiens | 35 | ALA1138619 | cell-based format | Scientific Literature | |
13. | ALA1048405 | B | Inhibition of human autotaxin isolated from MDA-MB-231 cells assessed as blockade of FS3 substrate hydrolysis by FRET assay | Homo sapiens | 16 | ALA1154760 | cell-based format | Scientific Literature | |
14. | ALA1048406 | B | Inhibition of human autotaxin isolated from MDA-MB-231 cells assessed as FS3 substrate hydrolysis at 10 uM by FRET assay | Homo sapiens | 31 | ALA1154760 | cell-based format | Scientific Literature | |
15. | ALA1048407 | B | Competitive inhibition of human autotaxin at free state isolated from MDA-MB-231 cells assessed as blockade of FS3 substrate hydrolysis by FRET assay | Homo sapiens | 7 | ALA1154760 | cell-based format | Scientific Literature | |
16. | ALA1048408 | B | Noncompetitive type inhibition of human autotaxin at enzyme-substrate complex isolated from MDA-MB-231 cells assessed as blockade of FS3 substrate hydrolysis by FRET assay | Homo sapiens | 1 | ALA1154760 | cell-based format | Scientific Literature | |
17. | ALA1048411 | B | Mixed type inhibition of human autotaxin at free state isolated from MDA-MB-231 cells assessed as blockade of FS3 substrate hydrolysis by FRET assay | Homo sapiens | 4 | ALA1154760 | cell-based format | Scientific Literature | |
18. | ALA1048412 | B | Noncompetitive type inhibition of human autotaxin at free state isolated from MDA-MB-231 cells assessed as blockade of FS3 substrate hydrolysis by FRET assay | Homo sapiens | 3 | ALA1154760 | cell-based format | Scientific Literature | |
19. | ALA1048413 | B | Mixed type inhibition of human autotaxin at enzyme-substrate complex isolated from MDA-MB-231 cells assessed as blockade of FS3 substrate hydrolysis by FRET assay | Homo sapiens | 4 | ALA1154760 | cell-based format | Scientific Literature | |
20. | ALA1066425 | B | Inhibition of autotaxin-mediated FS3 hydrolysis in human MDA-MB-435 cells at 10 uM by amplex red protocol | Homo sapiens | 7 | ALA1157718 | cell-based format | Scientific Literature |