| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA2090271 | B | Inhibition of human recombinant KLK7 expressed in insect cell/baculovirus using Abz-KLYSSKQ-EDDnp as substrate by FRET analysis | Homo sapiens | 5 | assay format | Scientific Literature | ||
| 2. | ALA2090272 | B | Reversible competitive inhibition of recombinant human KLK7 expressed in insect cell/baculovirus using Abz-KLYSSKQ-EDDnp as substrate by Eadie-Hofstee plot analysis | Homo sapiens | 2 | assay format | Scientific Literature | ||
| 3. | ALA2090273 | B | Competitive inhibition of recombinant human KLK7 expressed in insect cell/baculovirus using Abz-KLYSSKQ-EDDnp as substrate by Dixon plot analysis | Homo sapiens | 5 | assay format | Scientific Literature | ||
| 4. | ALA1837531 | B | Inhibition of human kallikrein 7 using Abz-KLYSSKQ-EDDnp as substrate by spectrofluorimetric assay | Homo sapiens | 3 | single protein format | Scientific Literature | ||
| 5. | ALA1837532 | B | Inhibition of human kallikrein 7 using Abz-KLYSSKQ-EDDnp as substrate by Lineweaver-Burk plot analysis | Homo sapiens | 3 | single protein format | Scientific Literature | ||
| 6. | ALA1837534 | B | Competitive inhibition of human kallikrein 7 using Abz-KLYSSKQ-EDDnp as substrate by Lineweaver-Burk plot analysis | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 7. | ALA2412634 | B | Binding affinity to human kallikrein 7 assessed as half life of deacylated enzyme | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 8. | ALA2412636 | B | Binding affinity to human kallikrein 7 assessed as deacylation of enzyme relative to control | Homo sapiens | 3 | single protein format | Scientific Literature | ||
| 9. | ALA2412641 | B | Inhibition of human kallikrein 7 at 296 nM to 1 uM at pH 8 by fluorescence assay | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 10. | ALA2412642 | B | Inhibition of human kallikrein 7 at 0.5 to 8 uM at pH 8 by fluorescence assay | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 11. | ALA2412649 | B | Inhibition of human kallikrein 7 measured after 15 mins at pH 8 by fluorescence assay | Homo sapiens | 7 | single protein format | Scientific Literature | ||
| 12. | ALA3100741 | B | Ratio of Ki for mixed-type inhibition of human kallikrein7 assessed as enzyme-substrate-inhibitor complex to Ki for mixed-type inhibition of human kallikrein7 assessed as enzyme-inhibitor complex | Homo sapiens | 8 | single protein format | Scientific Literature | ||
| 13. | ALA3100742 | B | Mixed-type inhibition of human kallikrein7 using Suc-Leu-Leu-Val-Tyr-AMC as substrate assessed as enzyme-substrate-inhibitor complex after 15 to 60 mins by Lineweaver-Burk/Eadie-Hofstee plot analysis | Homo sapiens | 8 | single protein format | Scientific Literature | ||
| 14. | ALA3100743 | B | Mixed-type inhibition of human kallikrein7 using Suc-Leu-Leu-Val-Tyr-AMC as substrate assessed as enzyme-inhibitor complex after 15 to 60 mins by Lineweaver-Burk/Eadie-Hofstee plot analysis | Homo sapiens | 8 | single protein format | Scientific Literature | ||
| 15. | ALA3100874 | B | Reversible inhibition of human kallikrein7 using Suc-Leu-Leu-Val-Tyr-AMC as substrate after 15 to 60 mins by fluorescence assay | Homo sapiens | 16 | single protein format | Scientific Literature | ||
| 16. | ALA3100880 | B | Inhibition of human kallikrein7 using Suc-Leu-Leu-Val-Tyr-AMC as substrate at 50 uM after 15 mins by fluorescence assay | Homo sapiens | 8 | single protein format | Scientific Literature | ||
| 17. | ALA3100881 | B | Inhibition of human kallikrein7 using Suc-Leu-Leu-Val-Tyr-AMC as substrate after 15 mins by fluorescence assay | Homo sapiens | 8 | single protein format | Scientific Literature | ||
| 18. | ALA3110696 | B | Inhibition of human recombinant KLK7 expressed in baculovirus-infected insect cell system using Abz-KLYSSKQ-Eddnp as substrate incubated for 5 mins prior to substrate addition by FRET assay | Homo sapiens | 20 | assay format | Scientific Literature | ||
| 19. | ALA3110697 | B | Competitive inhibition of human recombinant KLK7 expressed in baculovirus-infected insect cell system using Abz-KLYSSKQ-Eddnp as substrate incubated for 5 mins prior to substrate addition by Lineweaver-Burk plot analysis | Homo sapiens | 20 | assay format | Scientific Literature | ||
| 20. | ALA3214851 | B | PubChem BioAssay. Fluorescence Intensity-based biochemical primary high throughput dose response assay to identify activators of kallikrein-7 (K7) zymogen. (Class of assay: confirmatory) | 248 | single protein format | PubChem BioAssays |
The page will load shortly, Thanks for your patience!